6-Azaspiro[2.5]octanes as small molecule agonists of the human glucagon-like peptide-1 receptor.

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Title: 6-Azaspiro[2.5]octanes as small molecule agonists of the human glucagon-like peptide-1 receptor.
Authors: Aspnes GE; Pfizer Medicine Design, Cambridge, MA 02139, United States., Bagley SW; Pfizer Medicine Design, Groton, CT 06340, United States., Coffey SB; Pfizer Medicine Design, Groton, CT 06340, United States., Conn EL; Pfizer Medicine Design, Groton, CT 06340, United States., Curto JM; Pfizer Medicine Design, Groton, CT 06340, United States., Edmonds DJ; Pfizer Medicine Design, Cambridge, MA 02139, United States., Genovino J; Pfizer Medicine Design, Groton, CT 06340, United States., Griffith DA; Pfizer Medicine Design, Cambridge, MA 02139, United States., Ingle G; Pfizer Medicine Design, Groton, CT 06340, United States., Jiao W; Pfizer Medicine Design, Groton, CT 06340, United States., Limberakis C; Pfizer Medicine Design, Groton, CT 06340, United States., Mathiowetz AM; Pfizer Medicine Design, Cambridge, MA 02139, United States., Piotrowski DW; Pfizer Medicine Design, Groton, CT 06340, United States. Electronic address: david.w.piotrowski@comcast.net., Rose CR; Pfizer Medicine Design, Groton, CT 06340, United States., Ruggeri RB; Pfizer Medicine Design, Cambridge, MA 02139, United States., Wei L; Pfizer Medicine Design, Groton, CT 06340, United States.
Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2023 Oct 01; Vol. 94, pp. 129454. Date of Electronic Publication: 2023 Aug 15.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: 6-Azaspiro[2.5]octanes as small molecule agonists of the human glucagon-like peptide-1 receptor.
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  Data: <searchLink fieldCode="AU" term="%22Aspnes+GE%22">Aspnes GE</searchLink>; Pfizer Medicine Design, Cambridge, MA 02139, United States.<br /><searchLink fieldCode="AU" term="%22Bagley+SW%22">Bagley SW</searchLink>; Pfizer Medicine Design, Groton, CT 06340, United States.<br /><searchLink fieldCode="AU" term="%22Coffey+SB%22">Coffey SB</searchLink>; Pfizer Medicine Design, Groton, CT 06340, United States.<br /><searchLink fieldCode="AU" term="%22Conn+EL%22">Conn EL</searchLink>; Pfizer Medicine Design, Groton, CT 06340, United States.<br /><searchLink fieldCode="AU" term="%22Curto+JM%22">Curto JM</searchLink>; Pfizer Medicine Design, Groton, CT 06340, United States.<br /><searchLink fieldCode="AU" term="%22Edmonds+DJ%22">Edmonds DJ</searchLink>; Pfizer Medicine Design, Cambridge, MA 02139, United States.<br /><searchLink fieldCode="AU" term="%22Genovino+J%22">Genovino J</searchLink>; Pfizer Medicine Design, Groton, CT 06340, United States.<br /><searchLink fieldCode="AU" term="%22Griffith+DA%22">Griffith DA</searchLink>; Pfizer Medicine Design, Cambridge, MA 02139, United States.<br /><searchLink fieldCode="AU" term="%22Ingle+G%22">Ingle G</searchLink>; Pfizer Medicine Design, Groton, CT 06340, United States.<br /><searchLink fieldCode="AU" term="%22Jiao+W%22">Jiao W</searchLink>; Pfizer Medicine Design, Groton, CT 06340, United States.<br /><searchLink fieldCode="AU" term="%22Limberakis+C%22">Limberakis C</searchLink>; Pfizer Medicine Design, Groton, CT 06340, United States.<br /><searchLink fieldCode="AU" term="%22Mathiowetz+AM%22">Mathiowetz AM</searchLink>; Pfizer Medicine Design, Cambridge, MA 02139, United States.<br /><searchLink fieldCode="AU" term="%22Piotrowski+DW%22">Piotrowski DW</searchLink>; Pfizer Medicine Design, Groton, CT 06340, United States. Electronic address: david.w.piotrowski@comcast.net.<br /><searchLink fieldCode="AU" term="%22Rose+CR%22">Rose CR</searchLink>; Pfizer Medicine Design, Groton, CT 06340, United States.<br /><searchLink fieldCode="AU" term="%22Ruggeri+RB%22">Ruggeri RB</searchLink>; Pfizer Medicine Design, Cambridge, MA 02139, United States.<br /><searchLink fieldCode="AU" term="%22Wei+L%22">Wei L</searchLink>; Pfizer Medicine Design, Groton, CT 06340, United States.
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  Data: <searchLink fieldCode="JN" term="%229107377%22">Bioorganic & medicinal chemistry letters</searchLink> [Bioorg Med Chem Lett] 2023 Oct 01; Vol. 94, pp. 129454. <i>Date of Electronic Publication: </i>2023 Aug 15.
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