Piperacetazine Directly Binds to the PAX3::FOXO1 Fusion Protein and Inhibits Its Transcriptional Activity.

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Title: Piperacetazine Directly Binds to the PAX3::FOXO1 Fusion Protein and Inhibits Its Transcriptional Activity.
Authors: Nakazawa K; Department of Oncology, Georgetown University Medical Center, Georgetown University, Washington, District of Columbia., Shaw T; Department of Oncology, Georgetown University Medical Center, Georgetown University, Washington, District of Columbia., Song YK; Genetics Branch, Center for Cancer Research, NCI, NIH, Bethesda, Maryland., Kouassi-Brou M; Department of Oncology, Georgetown University Medical Center, Georgetown University, Washington, District of Columbia., Molotkova A; Department of Oncology, Georgetown University Medical Center, Georgetown University, Washington, District of Columbia., Tiwari PB; Department of Oncology, Georgetown University Medical Center, Georgetown University, Washington, District of Columbia., Chou HC; Genetics Branch, Center for Cancer Research, NCI, NIH, Bethesda, Maryland., Wen X; Genetics Branch, Center for Cancer Research, NCI, NIH, Bethesda, Maryland., Wei JS; Genetics Branch, Center for Cancer Research, NCI, NIH, Bethesda, Maryland., Deniz E; Department of Oncology, Georgetown University Medical Center, Georgetown University, Washington, District of Columbia., Toretsky JA; Department of Oncology, Georgetown University Medical Center, Georgetown University, Washington, District of Columbia., Keller C; Children's Cancer Therapy Development Institute, Hillsboro, Oregon., Barr FG; Laboratory of Pathology, Center for Cancer Research, NCI, Bethesda, Maryland., Khan J; Genetics Branch, Center for Cancer Research, NCI, NIH, Bethesda, Maryland., Üren A; Department of Oncology, Georgetown University Medical Center, Georgetown University, Washington, District of Columbia.
Source: Cancer research communications [Cancer Res Commun] 2023 Oct 06; Vol. 3 (10), pp. 2030-2043.
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
Journal Info: Publisher: American Association for Cancer Research Country of Publication: United States NLM ID: 9918281580506676 Publication Model: Print Cited Medium: Internet ISSN: 2767-9764 (Electronic) Linking ISSN: 27679764 NLM ISO Abbreviation: Cancer Res Commun Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:2767-9764
DOI:10.1158/2767-9764.CRC-23-0119