Comparative Analysis of Drug-like EP300/CREBBP Acetyltransferase Inhibitors.

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Title: Comparative Analysis of Drug-like EP300/CREBBP Acetyltransferase Inhibitors.
Authors: Crawford MC; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States., Tripu DR; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States., Barritt SA; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, Massachusetts 02215, United States., Jing Y; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States., Gallimore D; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States., Kales SC; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States., Bhanu NV; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri 63110, United States., Xiong Y; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States., Fang Y; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States., Butler KAT; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States., LeClair CA; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States., Coussens NP; Molecular Pharmacology Laboratories, Applied and Developmental Research Directorate, Frederick National Laboratory for Cancer Research, Frederick, Maryland 21702, United States., Simeonov A; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States., Garcia BA; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri 63110, United States., Dibble CC; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, Massachusetts 02215, United States., Meier JL; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, Massachusetts 02215, United States.
Source: ACS chemical biology [ACS Chem Biol] 2023 Oct 20; Vol. 18 (10), pp. 2249-2258. Date of Electronic Publication: 2023 Sep 22.
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, N.I.H., Intramural; Research Support, Non-U.S. Gov't
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101282906 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1554-8937 (Electronic) Linking ISSN: 15548929 NLM ISO Abbreviation: ACS Chem Biol Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Comparative Analysis of Drug-like EP300/CREBBP Acetyltransferase Inhibitors.
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  Data: <searchLink fieldCode="AU" term="%22Crawford+MC%22">Crawford MC</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States.<br /><searchLink fieldCode="AU" term="%22Tripu+DR%22">Tripu DR</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States.<br /><searchLink fieldCode="AU" term="%22Barritt+SA%22">Barritt SA</searchLink>; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, Massachusetts 02215, United States.<br /><searchLink fieldCode="AU" term="%22Jing+Y%22">Jing Y</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States.<br /><searchLink fieldCode="AU" term="%22Gallimore+D%22">Gallimore D</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States.<br /><searchLink fieldCode="AU" term="%22Kales+SC%22">Kales SC</searchLink>; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States.<br /><searchLink fieldCode="AU" term="%22Bhanu+NV%22">Bhanu NV</searchLink>; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri 63110, United States.<br /><searchLink fieldCode="AU" term="%22Xiong+Y%22">Xiong Y</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States.<br /><searchLink fieldCode="AU" term="%22Fang+Y%22">Fang Y</searchLink>; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States.<br /><searchLink fieldCode="AU" term="%22Butler+KAT%22">Butler KAT</searchLink>; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States.<br /><searchLink fieldCode="AU" term="%22LeClair+CA%22">LeClair CA</searchLink>; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States.<br /><searchLink fieldCode="AU" term="%22Coussens+NP%22">Coussens NP</searchLink>; Molecular Pharmacology Laboratories, Applied and Developmental Research Directorate, Frederick National Laboratory for Cancer Research, Frederick, Maryland 21702, United States.<br /><searchLink fieldCode="AU" term="%22Simeonov+A%22">Simeonov A</searchLink>; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States.<br /><searchLink fieldCode="AU" term="%22Garcia+BA%22">Garcia BA</searchLink>; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri 63110, United States.<br /><searchLink fieldCode="AU" term="%22Dibble+CC%22">Dibble CC</searchLink>; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, Massachusetts 02215, United States.<br /><searchLink fieldCode="AU" term="%22Meier+JL%22">Meier JL</searchLink>; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, Massachusetts 02215, United States.
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  Data: <searchLink fieldCode="JN" term="%22101282906%22">ACS chemical biology</searchLink> [ACS Chem Biol] 2023 Oct 20; Vol. 18 (10), pp. 2249-2258. <i>Date of Electronic Publication: </i>2023 Sep 22.
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        Value: 10.1021/acschembio.3c00293
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              Text: 2023 Oct 20
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