Comparative Analysis of Drug-like EP300/CREBBP Acetyltransferase Inhibitors.
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| Title: | Comparative Analysis of Drug-like EP300/CREBBP Acetyltransferase Inhibitors. |
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| Authors: | Crawford MC; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States., Tripu DR; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States., Barritt SA; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, Massachusetts 02215, United States., Jing Y; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States., Gallimore D; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States., Kales SC; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States., Bhanu NV; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri 63110, United States., Xiong Y; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States., Fang Y; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States., Butler KAT; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States., LeClair CA; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States., Coussens NP; Molecular Pharmacology Laboratories, Applied and Developmental Research Directorate, Frederick National Laboratory for Cancer Research, Frederick, Maryland 21702, United States., Simeonov A; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States., Garcia BA; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri 63110, United States., Dibble CC; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, Massachusetts 02215, United States., Meier JL; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, Massachusetts 02215, United States. |
| Source: | ACS chemical biology [ACS Chem Biol] 2023 Oct 20; Vol. 18 (10), pp. 2249-2258. Date of Electronic Publication: 2023 Sep 22. |
| Publication Type: | Journal Article; Research Support, N.I.H., Extramural; Research Support, N.I.H., Intramural; Research Support, Non-U.S. Gov't |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 101282906 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1554-8937 (Electronic) Linking ISSN: 15548929 NLM ISO Abbreviation: ACS Chem Biol Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 37737090 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Comparative Analysis of Drug-like EP300/CREBBP Acetyltransferase Inhibitors. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Crawford+MC%22">Crawford MC</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States.<br /><searchLink fieldCode="AU" term="%22Tripu+DR%22">Tripu DR</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States.<br /><searchLink fieldCode="AU" term="%22Barritt+SA%22">Barritt SA</searchLink>; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, Massachusetts 02215, United States.<br /><searchLink fieldCode="AU" term="%22Jing+Y%22">Jing Y</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States.<br /><searchLink fieldCode="AU" term="%22Gallimore+D%22">Gallimore D</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States.<br /><searchLink fieldCode="AU" term="%22Kales+SC%22">Kales SC</searchLink>; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States.<br /><searchLink fieldCode="AU" term="%22Bhanu+NV%22">Bhanu NV</searchLink>; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri 63110, United States.<br /><searchLink fieldCode="AU" term="%22Xiong+Y%22">Xiong Y</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States.<br /><searchLink fieldCode="AU" term="%22Fang+Y%22">Fang Y</searchLink>; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States.<br /><searchLink fieldCode="AU" term="%22Butler+KAT%22">Butler KAT</searchLink>; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States.<br /><searchLink fieldCode="AU" term="%22LeClair+CA%22">LeClair CA</searchLink>; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States.<br /><searchLink fieldCode="AU" term="%22Coussens+NP%22">Coussens NP</searchLink>; Molecular Pharmacology Laboratories, Applied and Developmental Research Directorate, Frederick National Laboratory for Cancer Research, Frederick, Maryland 21702, United States.<br /><searchLink fieldCode="AU" term="%22Simeonov+A%22">Simeonov A</searchLink>; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, United States.<br /><searchLink fieldCode="AU" term="%22Garcia+BA%22">Garcia BA</searchLink>; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri 63110, United States.<br /><searchLink fieldCode="AU" term="%22Dibble+CC%22">Dibble CC</searchLink>; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, Massachusetts 02215, United States.<br /><searchLink fieldCode="AU" term="%22Meier+JL%22">Meier JL</searchLink>; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, Massachusetts 02215, United States. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101282906%22">ACS chemical biology</searchLink> [ACS Chem Biol] 2023 Oct 20; Vol. 18 (10), pp. 2249-2258. <i>Date of Electronic Publication: </i>2023 Sep 22. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article; Research Support, N.I.H., Extramural; Research Support, N.I.H., Intramural; Research Support, Non-U.S. Gov't – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101282906 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1554-8937 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2215548929%22">15548929 </searchLink><i>NLM ISO Abbreviation: </i>ACS Chem Biol <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=37737090 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/acschembio.3c00293 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 2249 Titles: – TitleFull: Comparative Analysis of Drug-like EP300/CREBBP Acetyltransferase Inhibitors. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Crawford MC – PersonEntity: Name: NameFull: Tripu DR – PersonEntity: Name: NameFull: Barritt SA – PersonEntity: Name: NameFull: Jing Y – PersonEntity: Name: NameFull: Gallimore D – PersonEntity: Name: NameFull: Kales SC – PersonEntity: Name: NameFull: Bhanu NV – PersonEntity: Name: NameFull: Xiong Y – PersonEntity: Name: NameFull: Fang Y – PersonEntity: Name: NameFull: Butler KAT – PersonEntity: Name: NameFull: LeClair CA – PersonEntity: Name: NameFull: Coussens NP – PersonEntity: Name: NameFull: Simeonov A – PersonEntity: Name: NameFull: Garcia BA – PersonEntity: Name: NameFull: Dibble CC – PersonEntity: Name: NameFull: Meier JL IsPartOfRelationships: – BibEntity: Dates: – D: 20 M: 10 Text: 2023 Oct 20 Type: published Y: 2023 Identifiers: – Type: issn-electronic Value: 1554-8937 Numbering: – Type: volume Value: 18 – Type: issue Value: 10 Titles: – TitleFull: ACS chemical biology Type: main |
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