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Discovery of a novel series of selective macrocyclic PKCTheta inhibitors.

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Title: Discovery of a novel series of selective macrocyclic PKCTheta inhibitors.
Authors: Crosignani S; Galderma SA, Av. d'Ouchy 4, 1006 Lausanne, Switzerland. Electronic address: stefano.crosignani@gmail.com., Campos S; Pharmaron Discovery & Early Development, West Hill Innovation Park, Hertford Road, Hoddesdon, Hertfordshire EN11 9FH, UK., Bouix-Peter C; Galderma SA, Av. d'Ouchy 4, 1006 Lausanne, Switzerland., Harris C; Galderma SA, Av. d'Ouchy 4, 1006 Lausanne, Switzerland., Talbot E; Pharmaron Discovery & Early Development, West Hill Innovation Park, Hertford Road, Hoddesdon, Hertfordshire EN11 9FH, UK., Hu H; Pharmaron Discovery & Early Development, West Hill Innovation Park, Hertford Road, Hoddesdon, Hertfordshire EN11 9FH, UK., Wang S; Pharmaron Discovery & Early Development, West Hill Innovation Park, Hertford Road, Hoddesdon, Hertfordshire EN11 9FH, UK., Maclean J; Pharmaron Discovery & Early Development, West Hill Innovation Park, Hertford Road, Hoddesdon, Hertfordshire EN11 9FH, UK., Zanelli U; Galderma SA, Av. d'Ouchy 4, 1006 Lausanne, Switzerland., Taylor S; Pharmaron Discovery & Early Development, West Hill Innovation Park, Hertford Road, Hoddesdon, Hertfordshire EN11 9FH, UK., Foote K; Pharmaron Discovery & Early Development, West Hill Innovation Park, Hertford Road, Hoddesdon, Hertfordshire EN11 9FH, UK., Hacini-Rachinel F; Galderma SA, Av. d'Ouchy 4, 1006 Lausanne, Switzerland., Nicodeme E; Galderma SA, Av. d'Ouchy 4, 1006 Lausanne, Switzerland., Julia V; Galderma SA, Av. d'Ouchy 4, 1006 Lausanne, Switzerland.
Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2024 Mar 01; Vol. 100, pp. 129630. Date of Electronic Publication: 2024 Feb 01.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE; PubMed not MEDLINE
Database: MEDLINE Ultimate
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  Data: Discovery of a novel series of selective macrocyclic PKCTheta inhibitors.
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  Data: <searchLink fieldCode="AU" term="%22Crosignani+S%22">Crosignani S</searchLink>; Galderma SA, Av. d'Ouchy 4, 1006 Lausanne, Switzerland. Electronic address: stefano.crosignani@gmail.com.<br /><searchLink fieldCode="AU" term="%22Campos+S%22">Campos S</searchLink>; Pharmaron Discovery & Early Development, West Hill Innovation Park, Hertford Road, Hoddesdon, Hertfordshire EN11 9FH, UK.<br /><searchLink fieldCode="AU" term="%22Bouix-Peter+C%22">Bouix-Peter C</searchLink>; Galderma SA, Av. d'Ouchy 4, 1006 Lausanne, Switzerland.<br /><searchLink fieldCode="AU" term="%22Harris+C%22">Harris C</searchLink>; Galderma SA, Av. d'Ouchy 4, 1006 Lausanne, Switzerland.<br /><searchLink fieldCode="AU" term="%22Talbot+E%22">Talbot E</searchLink>; Pharmaron Discovery & Early Development, West Hill Innovation Park, Hertford Road, Hoddesdon, Hertfordshire EN11 9FH, UK.<br /><searchLink fieldCode="AU" term="%22Hu+H%22">Hu H</searchLink>; Pharmaron Discovery & Early Development, West Hill Innovation Park, Hertford Road, Hoddesdon, Hertfordshire EN11 9FH, UK.<br /><searchLink fieldCode="AU" term="%22Wang+S%22">Wang S</searchLink>; Pharmaron Discovery & Early Development, West Hill Innovation Park, Hertford Road, Hoddesdon, Hertfordshire EN11 9FH, UK.<br /><searchLink fieldCode="AU" term="%22Maclean+J%22">Maclean J</searchLink>; Pharmaron Discovery & Early Development, West Hill Innovation Park, Hertford Road, Hoddesdon, Hertfordshire EN11 9FH, UK.<br /><searchLink fieldCode="AU" term="%22Zanelli+U%22">Zanelli U</searchLink>; Galderma SA, Av. d'Ouchy 4, 1006 Lausanne, Switzerland.<br /><searchLink fieldCode="AU" term="%22Taylor+S%22">Taylor S</searchLink>; Pharmaron Discovery & Early Development, West Hill Innovation Park, Hertford Road, Hoddesdon, Hertfordshire EN11 9FH, UK.<br /><searchLink fieldCode="AU" term="%22Foote+K%22">Foote K</searchLink>; Pharmaron Discovery & Early Development, West Hill Innovation Park, Hertford Road, Hoddesdon, Hertfordshire EN11 9FH, UK.<br /><searchLink fieldCode="AU" term="%22Hacini-Rachinel+F%22">Hacini-Rachinel F</searchLink>; Galderma SA, Av. d'Ouchy 4, 1006 Lausanne, Switzerland.<br /><searchLink fieldCode="AU" term="%22Nicodeme+E%22">Nicodeme E</searchLink>; Galderma SA, Av. d'Ouchy 4, 1006 Lausanne, Switzerland.<br /><searchLink fieldCode="AU" term="%22Julia+V%22">Julia V</searchLink>; Galderma SA, Av. d'Ouchy 4, 1006 Lausanne, Switzerland.
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  Data: <searchLink fieldCode="JN" term="%229107377%22">Bioorganic & medicinal chemistry letters</searchLink> [Bioorg Med Chem Lett] 2024 Mar 01; Vol. 100, pp. 129630. <i>Date of Electronic Publication: </i>2024 Feb 01.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Science+Ltd%22">Elsevier Science Ltd </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>9107377 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1464-3405 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%220960894X%22">0960894X </searchLink><i>NLM ISO Abbreviation: </i>Bioorg Med Chem Lett <i>Subsets: </i>MEDLINE; PubMed not MEDLINE
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              Text: 2024 Mar 01
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