Novel modifications of PARP inhibitor veliparib increase PARP1 binding to DNA breaks.

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Title: Novel modifications of PARP inhibitor veliparib increase PARP1 binding to DNA breaks.
Authors: Velagapudi UK; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, New York 11439, U.S.A., Rouleau-Turcotte É; Department of Biochemistry and Molecular Medicine, Université de Montréal, Montréal, Canada H3T 1J4., Billur R; Department of Biochemistry and Biophysics, Penn Center for Genome Integrity, Epigenetics Institute, Perelman School of Medicine, University of Pennsylvania, Philadelphia, PA 19104-6059, U.S.A., Shao X; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, New York 11439, U.S.A., Patil M; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, New York 11439, U.S.A., Black BE; Department of Biochemistry and Biophysics, Penn Center for Genome Integrity, Epigenetics Institute, Perelman School of Medicine, University of Pennsylvania, Philadelphia, PA 19104-6059, U.S.A., Pascal JM; Department of Biochemistry and Molecular Medicine, Université de Montréal, Montréal, Canada H3T 1J4., Talele TT; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, New York 11439, U.S.A.
Source: The Biochemical journal [Biochem J] 2024 Mar 20; Vol. 481 (6), pp. 437-460.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, N.I.H., Extramural
Journal Info: Publisher: Published by Portland Press on behalf of the Biochemical Society Country of Publication: England NLM ID: 2984726R Publication Model: Print Cited Medium: Internet ISSN: 1470-8728 (Electronic) Linking ISSN: 02646021 NLM ISO Abbreviation: Biochem J Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Novel modifications of PARP inhibitor veliparib increase PARP1 binding to DNA breaks.
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  Data: <searchLink fieldCode="AU" term="%22Velagapudi+UK%22">Velagapudi UK</searchLink>; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, New York 11439, U.S.A.<br /><searchLink fieldCode="AU" term="%22Rouleau-Turcotte+É%22">Rouleau-Turcotte É</searchLink>; Department of Biochemistry and Molecular Medicine, Université de Montréal, Montréal, Canada H3T 1J4.<br /><searchLink fieldCode="AU" term="%22Billur+R%22">Billur R</searchLink>; Department of Biochemistry and Biophysics, Penn Center for Genome Integrity, Epigenetics Institute, Perelman School of Medicine, University of Pennsylvania, Philadelphia, PA 19104-6059, U.S.A.<br /><searchLink fieldCode="AU" term="%22Shao+X%22">Shao X</searchLink>; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, New York 11439, U.S.A.<br /><searchLink fieldCode="AU" term="%22Patil+M%22">Patil M</searchLink>; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, New York 11439, U.S.A.<br /><searchLink fieldCode="AU" term="%22Black+BE%22">Black BE</searchLink>; Department of Biochemistry and Biophysics, Penn Center for Genome Integrity, Epigenetics Institute, Perelman School of Medicine, University of Pennsylvania, Philadelphia, PA 19104-6059, U.S.A.<br /><searchLink fieldCode="AU" term="%22Pascal+JM%22">Pascal JM</searchLink>; Department of Biochemistry and Molecular Medicine, Université de Montréal, Montréal, Canada H3T 1J4.<br /><searchLink fieldCode="AU" term="%22Talele+TT%22">Talele TT</searchLink>; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, New York 11439, U.S.A.
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  Data: <searchLink fieldCode="JN" term="%222984726R%22">The Biochemical journal</searchLink> [Biochem J] 2024 Mar 20; Vol. 481 (6), pp. 437-460.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Published+by+Portland+Press+on+behalf+of+the+Biochemical+Society%22">Published by Portland Press on behalf of the Biochemical Society </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>2984726R <i>Publication Model: </i>Print <i>Cited Medium: </i>Internet <i>ISSN: </i>1470-8728 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2202646021%22">02646021 </searchLink><i>NLM ISO Abbreviation: </i>Biochem J <i>Subsets: </i>MEDLINE
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        Value: 10.1042/BCJ20230406
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              Text: 2024 Mar 20
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