From Functional Fatty Acids to Potent and Selective Natural-Product-Inspired Mimetics via Conformational Profiling.

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Title: From Functional Fatty Acids to Potent and Selective Natural-Product-Inspired Mimetics via Conformational Profiling.
Authors: Markham LE; Department of Chemistry, Dartmouth College, 6128 Burke Laboratory, Hanover, New Hampshire 03755, United States., Koelblen T; University of Florida Genetics Institute, P.O. Box 103610, 2033 Mowry Road, Gainesville, Florida 32610, United States., Chobanian HR; ROME Therapeutics, 201 Brookline Avenue, Suite 1001, Boston, Massachusetts 02215, United States., Follis AV; ROME Therapeutics, 201 Brookline Avenue, Suite 1001, Boston, Massachusetts 02215, United States., Burris TP; University of Florida Genetics Institute, P.O. Box 103610, 2033 Mowry Road, Gainesville, Florida 32610, United States., Micalizio GC; Department of Chemistry, Dartmouth College, 6128 Burke Laboratory, Hanover, New Hampshire 03755, United States.
Source: ACS central science [ACS Cent Sci] 2024 Feb 12; Vol. 10 (2), pp. 477-486. Date of Electronic Publication: 2024 Feb 12 (Print Publication: 2024).
Publication Type: Journal Article
Journal Info: Publisher: ACS Publications Country of Publication: United States NLM ID: 101660035 Publication Model: eCollection Cited Medium: Print ISSN: 2374-7943 (Print) Linking ISSN: 23747943 NLM ISO Abbreviation: ACS Cent Sci Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
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  Data: <searchLink fieldCode="AU" term="%22Markham+LE%22">Markham LE</searchLink>; Department of Chemistry, Dartmouth College, 6128 Burke Laboratory, Hanover, New Hampshire 03755, United States.<br /><searchLink fieldCode="AU" term="%22Koelblen+T%22">Koelblen T</searchLink>; University of Florida Genetics Institute, P.O. Box 103610, 2033 Mowry Road, Gainesville, Florida 32610, United States.<br /><searchLink fieldCode="AU" term="%22Chobanian+HR%22">Chobanian HR</searchLink>; ROME Therapeutics, 201 Brookline Avenue, Suite 1001, Boston, Massachusetts 02215, United States.<br /><searchLink fieldCode="AU" term="%22Follis+AV%22">Follis AV</searchLink>; ROME Therapeutics, 201 Brookline Avenue, Suite 1001, Boston, Massachusetts 02215, United States.<br /><searchLink fieldCode="AU" term="%22Burris+TP%22">Burris TP</searchLink>; University of Florida Genetics Institute, P.O. Box 103610, 2033 Mowry Road, Gainesville, Florida 32610, United States.<br /><searchLink fieldCode="AU" term="%22Micalizio+GC%22">Micalizio GC</searchLink>; Department of Chemistry, Dartmouth College, 6128 Burke Laboratory, Hanover, New Hampshire 03755, United States.
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        Value: 10.1021/acscentsci.3c01155
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