Liver-targeted polymeric prodrugs delivered subcutaneously improve tafenoquine therapeutic window for malaria radical cure.

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Title: Liver-targeted polymeric prodrugs delivered subcutaneously improve tafenoquine therapeutic window for malaria radical cure.
Authors: Pottenger AE; Department of Bioengineering, University of Washington, Seattle, WA 98195, USA., Roy D; Department of Bioengineering, University of Washington, Seattle, WA 98195, USA., Srinivasan S; Department of Bioengineering, University of Washington, Seattle, WA 98195, USA., Chavas TEJ; Department of Bioengineering, University of Washington, Seattle, WA 98195, USA., Vlaskin V; Department of Bioengineering, University of Washington, Seattle, WA 98195, USA., Ho DK; Department of Bioengineering, University of Washington, Seattle, WA 98195, USA., Livingston VC; Department of Bioengineering, University of Washington, Seattle, WA 98195, USA., Maktabi M; Department of Immunology and Microbiology, University of Colorado Anschutz School of Medicine, Aurora, CO 80045, USA., Lin H; Department of Drug Discovery, Experimental Therapeutics Branch, Walter Reed Army Institute of Research, Silver Spring, MD 20910, USA., Zhang J; Department of Drug Discovery, Experimental Therapeutics Branch, Walter Reed Army Institute of Research, Silver Spring, MD 20910, USA., Pybus B; Department of Drug Discovery, Experimental Therapeutics Branch, Walter Reed Army Institute of Research, Silver Spring, MD 20910, USA., Kudyba K; Department of Drug Discovery, Experimental Therapeutics Branch, Walter Reed Army Institute of Research, Silver Spring, MD 20910, USA., Roth A; Department of Drug Discovery, Experimental Therapeutics Branch, Walter Reed Army Institute of Research, Silver Spring, MD 20910, USA., Senter P; Seagen, Bothell, WA 98021, USA., Tyson G; George Tyson Consulting, Los Altos Hills, CA 94022, USA.; Department of Chemical and Biomolecular Engineering, University of California, Berkeley, Berkeley, CA 94720, USA., Huber HE; BioTD Strategies LLC, 213 Abbey Ln., Lansdale, PA 19446, USA., Wesche D; Certara, Princeton, NJ 08540, USA., Rochford R; Department of Immunology and Microbiology, University of Colorado Anschutz School of Medicine, Aurora, CO 80045, USA., Burke PA; Department of Bioengineering, University of Washington, Seattle, WA 98195, USA.; Burke Bioventures LLC, 1 Broadway 14th Floor, Cambridge, MA 02142, USA., Stayton PS; Department of Bioengineering, University of Washington, Seattle, WA 98195, USA.
Source: Science advances [Sci Adv] 2024 Apr 19; Vol. 10 (16), pp. eadk4492. Date of Electronic Publication: 2024 Apr 19.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: American Association for the Advancement of Science Country of Publication: United States NLM ID: 101653440 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2375-2548 (Electronic) Linking ISSN: 23752548 NLM ISO Abbreviation: Sci Adv Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:2375-2548
DOI:10.1126/sciadv.adk4492