Label-free detection of prostaglandin transporter (SLCO2A1) function and inhibition: insights by wound healing and TRACT assays.

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Title: Label-free detection of prostaglandin transporter (SLCO2A1) function and inhibition: insights by wound healing and TRACT assays.
Authors: Mocking TAM; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Leiden, Netherlands., van Oostveen WM; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Leiden, Netherlands.; Department of Rheumatology, Leiden University Medical Center, Leiden University, Leiden, Netherlands.; Immunology and Respiratory Diseases, Boehringer-Ingelheim, Ridgefield, CT, United States.; Oncode Institute, Leiden, Netherlands., van Veldhoven JPD; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Leiden, Netherlands.; Department of Rheumatology, Leiden University Medical Center, Leiden University, Leiden, Netherlands.; Immunology and Respiratory Diseases, Boehringer-Ingelheim, Ridgefield, CT, United States.; Oncode Institute, Leiden, Netherlands., Minnee H; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Leiden, Netherlands., Fehres CM; Department of Rheumatology, Leiden University Medical Center, Leiden University, Leiden, Netherlands., Whitehurst CE; Immunology and Respiratory Diseases, Boehringer-Ingelheim, Ridgefield, CT, United States., IJzerman AP; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Leiden, Netherlands., Heitman LH; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Leiden, Netherlands.; Oncode Institute, Leiden, Netherlands.
Source: Frontiers in pharmacology [Front Pharmacol] 2024 May 09; Vol. 15, pp. 1372109. Date of Electronic Publication: 2024 May 09 (Print Publication: 2024).
Publication Type: Journal Article
Journal Info: Publisher: Frontiers Media] Country of Publication: Switzerland NLM ID: 101548923 Publication Model: eCollection Cited Medium: Print ISSN: 1663-9812 (Print) Linking ISSN: 16639812 NLM ISO Abbreviation: Front Pharmacol Subsets: PubMed not MEDLINE
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  Data: Label-free detection of prostaglandin transporter (SLCO2A1) function and inhibition: insights by wound healing and TRACT assays.
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  Data: <searchLink fieldCode="AU" term="%22Mocking+TAM%22">Mocking TAM</searchLink>; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Leiden, Netherlands.<br /><searchLink fieldCode="AU" term="%22van+Oostveen+WM%22">van Oostveen WM</searchLink>; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Leiden, Netherlands.; Department of Rheumatology, Leiden University Medical Center, Leiden University, Leiden, Netherlands.; Immunology and Respiratory Diseases, Boehringer-Ingelheim, Ridgefield, CT, United States.; Oncode Institute, Leiden, Netherlands.<br /><searchLink fieldCode="AU" term="%22van+Veldhoven+JPD%22">van Veldhoven JPD</searchLink>; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Leiden, Netherlands.; Department of Rheumatology, Leiden University Medical Center, Leiden University, Leiden, Netherlands.; Immunology and Respiratory Diseases, Boehringer-Ingelheim, Ridgefield, CT, United States.; Oncode Institute, Leiden, Netherlands.<br /><searchLink fieldCode="AU" term="%22Minnee+H%22">Minnee H</searchLink>; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Leiden, Netherlands.<br /><searchLink fieldCode="AU" term="%22Fehres+CM%22">Fehres CM</searchLink>; Department of Rheumatology, Leiden University Medical Center, Leiden University, Leiden, Netherlands.<br /><searchLink fieldCode="AU" term="%22Whitehurst+CE%22">Whitehurst CE</searchLink>; Immunology and Respiratory Diseases, Boehringer-Ingelheim, Ridgefield, CT, United States.<br /><searchLink fieldCode="AU" term="%22IJzerman+AP%22">IJzerman AP</searchLink>; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Leiden, Netherlands.<br /><searchLink fieldCode="AU" term="%22Heitman+LH%22">Heitman LH</searchLink>; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, Leiden, Netherlands.; Oncode Institute, Leiden, Netherlands.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Frontiers+Media]%22">Frontiers Media] </searchLink><i>Country of Publication: </i>Switzerland <i>NLM ID: </i>101548923 <i>Publication Model: </i>eCollection <i>Cited Medium: </i>Print <i>ISSN: </i>1663-9812 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2216639812%22">16639812 </searchLink><i>NLM ISO Abbreviation: </i>Front Pharmacol <i>Subsets: </i>PubMed not MEDLINE
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        Value: 10.3389/fphar.2024.1372109
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      – TitleFull: Label-free detection of prostaglandin transporter (SLCO2A1) function and inhibition: insights by wound healing and TRACT assays.
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              Text: 2024 May 09
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