Minimal Involvement of P-gp and BCRP in Oral Absorption of Ensitrelvir, An Oral SARS-CoV-2 3C-like Protease Inhibitor, in a Non-Clinical Investigation.

Saved in:
Bibliographic Details
Title: Minimal Involvement of P-gp and BCRP in Oral Absorption of Ensitrelvir, An Oral SARS-CoV-2 3C-like Protease Inhibitor, in a Non-Clinical Investigation.
Authors: Watari R; Laboratory for Drug Discovery and Development, Shionogi & Co., Ltd.. Electronic address: ryosuke.watari@shionogi.co.jp., Tamura N; Laboratory for Drug Discovery and Development, Shionogi & Co., Ltd., Yoshida S; Laboratory for Drug Discovery and Development, Shionogi & Co., Ltd., Kido Y; Laboratory for Drug Discovery and Development, Shionogi & Co., Ltd., Matsuzaki T; Laboratory for Drug Discovery and Development, Shionogi & Co., Ltd.
Source: Journal of pharmaceutical sciences [J Pharm Sci] 2024 Sep; Vol. 113 (9), pp. 2871-2878. Date of Electronic Publication: 2024 Jun 15.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Country of Publication: United States NLM ID: 2985195R Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-6017 (Electronic) Linking ISSN: 00223549 NLM ISO Abbreviation: J Pharm Sci Subsets: MEDLINE
Database: MEDLINE Ultimate
FullText Text:
  Availability: 0
Header DbId: mdl
DbLabel: MEDLINE Ultimate
An: 38885812
AccessLevel: 2
PubType: Academic Journal
PubTypeId: academicJournal
PreciseRelevancyScore: 0
IllustrationInfo
Items – Name: Title
  Label: Title
  Group: Ti
  Data: Minimal Involvement of P-gp and BCRP in Oral Absorption of Ensitrelvir, An Oral SARS-CoV-2 3C-like Protease Inhibitor, in a Non-Clinical Investigation.
– Name: Author
  Label: Authors
  Group: Au
  Data: <searchLink fieldCode="AU" term="%22Watari+R%22">Watari R</searchLink>; Laboratory for Drug Discovery and Development, Shionogi & Co., Ltd.. Electronic address: ryosuke.watari@shionogi.co.jp.<br /><searchLink fieldCode="AU" term="%22Tamura+N%22">Tamura N</searchLink>; Laboratory for Drug Discovery and Development, Shionogi & Co., Ltd.<br /><searchLink fieldCode="AU" term="%22Yoshida+S%22">Yoshida S</searchLink>; Laboratory for Drug Discovery and Development, Shionogi & Co., Ltd.<br /><searchLink fieldCode="AU" term="%22Kido+Y%22">Kido Y</searchLink>; Laboratory for Drug Discovery and Development, Shionogi & Co., Ltd.<br /><searchLink fieldCode="AU" term="%22Matsuzaki+T%22">Matsuzaki T</searchLink>; Laboratory for Drug Discovery and Development, Shionogi & Co., Ltd.
– Name: TitleSource
  Label: Source
  Group: Src
  Data: <searchLink fieldCode="JN" term="%222985195R%22">Journal of pharmaceutical sciences</searchLink> [J Pharm Sci] 2024 Sep; Vol. 113 (9), pp. 2871-2878. <i>Date of Electronic Publication: </i>2024 Jun 15.
– Name: TypePub
  Label: Publication Type
  Group: TypPub
  Data: Journal Article
– Name: TitleSource
  Label: Journal Info
  Group: Src
  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier%22">Elsevier </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>2985195R <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1520-6017 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200223549%22">00223549 </searchLink><i>NLM ISO Abbreviation: </i>J Pharm Sci <i>Subsets: </i>MEDLINE
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=38885812
RecordInfo BibRecord:
  BibEntity:
    Identifiers:
      – Type: doi
        Value: 10.1016/j.xphs.2024.06.009
    Languages:
      – Code: eng
        Text: English
    PhysicalDescription:
      Pagination:
        StartPage: 2871
    Titles:
      – TitleFull: Minimal Involvement of P-gp and BCRP in Oral Absorption of Ensitrelvir, An Oral SARS-CoV-2 3C-like Protease Inhibitor, in a Non-Clinical Investigation.
        Type: main
  BibRelationships:
    HasContributorRelationships:
      – PersonEntity:
          Name:
            NameFull: Watari R
      – PersonEntity:
          Name:
            NameFull: Tamura N
      – PersonEntity:
          Name:
            NameFull: Yoshida S
      – PersonEntity:
          Name:
            NameFull: Kido Y
      – PersonEntity:
          Name:
            NameFull: Matsuzaki T
    IsPartOfRelationships:
      – BibEntity:
          Dates:
            – D: 01
              M: 09
              Text: 2024 Sep
              Type: published
              Y: 2024
          Identifiers:
            – Type: issn-electronic
              Value: 1520-6017
          Numbering:
            – Type: volume
              Value: 113
            – Type: issue
              Value: 9
          Titles:
            – TitleFull: Journal of pharmaceutical sciences
              Type: main
ResultId 1