Relevance of G protein-coupled receptor (GPCR) dynamics for receptor activation, signalling bias and allosteric modulation.
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| Title: | Relevance of G protein-coupled receptor (GPCR) dynamics for receptor activation, signalling bias and allosteric modulation. |
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| Authors: | Lopez-Balastegui M; Research Programme on Biomedical Informatics (GRIB), Hospital del Mar Medical Research Institute & Pompeu Fabra University, Barcelona, Spain., Stepniewski TM; Research Programme on Biomedical Informatics (GRIB), Hospital del Mar Medical Research Institute & Pompeu Fabra University, Barcelona, Spain.; InterAx Biotech AG, Villigen, Switzerland., Kogut-Günthel MM; Leibniz Institute for Food Systems Biology at the Technical University of Munich, Freising, Germany., Di Pizio A; Leibniz Institute for Food Systems Biology at the Technical University of Munich, Freising, Germany.; Chair for Chemoinformatics and Protein Modelling, Department of Molecular Life Science, School of Science, Technical University of Munich, Freising, Germany., Rosenkilde MM; Department of Biomedical Sciences, Faculty of Health and Medical Sciences University of Copenhagen, København N, Denmark., Mao J; Huairou Research Center, Institute of Chemistry, Chinese Academy of Sciences, Beijing, China., Selent J; Research Programme on Biomedical Informatics (GRIB), Hospital del Mar Medical Research Institute & Pompeu Fabra University, Barcelona, Spain. |
| Source: | British journal of pharmacology [Br J Pharmacol] 2025 Jul; Vol. 182 (14), pp. 3211-3224. Date of Electronic Publication: 2024 Jul 08. |
| Publication Type: | Journal Article; Review |
| Journal Info: | Publisher: Wiley Country of Publication: England NLM ID: 7502536 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1476-5381 (Electronic) Linking ISSN: 00071188 NLM ISO Abbreviation: Br J Pharmacol Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 38978399 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Relevance of G protein-coupled receptor (GPCR) dynamics for receptor activation, signalling bias and allosteric modulation. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Lopez-Balastegui+M%22">Lopez-Balastegui M</searchLink>; Research Programme on Biomedical Informatics (GRIB), Hospital del Mar Medical Research Institute & Pompeu Fabra University, Barcelona, Spain.<br /><searchLink fieldCode="AU" term="%22Stepniewski+TM%22">Stepniewski TM</searchLink>; Research Programme on Biomedical Informatics (GRIB), Hospital del Mar Medical Research Institute & Pompeu Fabra University, Barcelona, Spain.; InterAx Biotech AG, Villigen, Switzerland.<br /><searchLink fieldCode="AU" term="%22Kogut-Günthel+MM%22">Kogut-Günthel MM</searchLink>; Leibniz Institute for Food Systems Biology at the Technical University of Munich, Freising, Germany.<br /><searchLink fieldCode="AU" term="%22Di+Pizio+A%22">Di Pizio A</searchLink>; Leibniz Institute for Food Systems Biology at the Technical University of Munich, Freising, Germany.; Chair for Chemoinformatics and Protein Modelling, Department of Molecular Life Science, School of Science, Technical University of Munich, Freising, Germany.<br /><searchLink fieldCode="AU" term="%22Rosenkilde+MM%22">Rosenkilde MM</searchLink>; Department of Biomedical Sciences, Faculty of Health and Medical Sciences University of Copenhagen, København N, Denmark.<br /><searchLink fieldCode="AU" term="%22Mao+J%22">Mao J</searchLink>; Huairou Research Center, Institute of Chemistry, Chinese Academy of Sciences, Beijing, China.<br /><searchLink fieldCode="AU" term="%22Selent+J%22">Selent J</searchLink>; Research Programme on Biomedical Informatics (GRIB), Hospital del Mar Medical Research Institute & Pompeu Fabra University, Barcelona, Spain. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%227502536%22">British journal of pharmacology</searchLink> [Br J Pharmacol] 2025 Jul; Vol. 182 (14), pp. 3211-3224. <i>Date of Electronic Publication: </i>2024 Jul 08. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article; Review – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Wiley%22">Wiley </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>7502536 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1476-5381 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200071188%22">00071188 </searchLink><i>NLM ISO Abbreviation: </i>Br J Pharmacol <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=38978399 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1111/bph.16495 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 3211 Titles: – TitleFull: Relevance of G protein-coupled receptor (GPCR) dynamics for receptor activation, signalling bias and allosteric modulation. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Lopez-Balastegui M – PersonEntity: Name: NameFull: Stepniewski TM – PersonEntity: Name: NameFull: Kogut-Günthel MM – PersonEntity: Name: NameFull: Di Pizio A – PersonEntity: Name: NameFull: Rosenkilde MM – PersonEntity: Name: NameFull: Mao J – PersonEntity: Name: NameFull: Selent J IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 07 Text: 2025 Jul Type: published Y: 2025 Identifiers: – Type: issn-electronic Value: 1476-5381 Numbering: – Type: volume Value: 182 – Type: issue Value: 14 Titles: – TitleFull: British journal of pharmacology Type: main |
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