Relevance of G protein-coupled receptor (GPCR) dynamics for receptor activation, signalling bias and allosteric modulation.

Saved in:
Bibliographic Details
Title: Relevance of G protein-coupled receptor (GPCR) dynamics for receptor activation, signalling bias and allosteric modulation.
Authors: Lopez-Balastegui M; Research Programme on Biomedical Informatics (GRIB), Hospital del Mar Medical Research Institute & Pompeu Fabra University, Barcelona, Spain., Stepniewski TM; Research Programme on Biomedical Informatics (GRIB), Hospital del Mar Medical Research Institute & Pompeu Fabra University, Barcelona, Spain.; InterAx Biotech AG, Villigen, Switzerland., Kogut-Günthel MM; Leibniz Institute for Food Systems Biology at the Technical University of Munich, Freising, Germany., Di Pizio A; Leibniz Institute for Food Systems Biology at the Technical University of Munich, Freising, Germany.; Chair for Chemoinformatics and Protein Modelling, Department of Molecular Life Science, School of Science, Technical University of Munich, Freising, Germany., Rosenkilde MM; Department of Biomedical Sciences, Faculty of Health and Medical Sciences University of Copenhagen, København N, Denmark., Mao J; Huairou Research Center, Institute of Chemistry, Chinese Academy of Sciences, Beijing, China., Selent J; Research Programme on Biomedical Informatics (GRIB), Hospital del Mar Medical Research Institute & Pompeu Fabra University, Barcelona, Spain.
Source: British journal of pharmacology [Br J Pharmacol] 2025 Jul; Vol. 182 (14), pp. 3211-3224. Date of Electronic Publication: 2024 Jul 08.
Publication Type: Journal Article; Review
Journal Info: Publisher: Wiley Country of Publication: England NLM ID: 7502536 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1476-5381 (Electronic) Linking ISSN: 00071188 NLM ISO Abbreviation: Br J Pharmacol Subsets: MEDLINE
Database: MEDLINE Ultimate
Full text is not displayed to guests.
FullText Links:
  – Type: pdflink
Text:
  Availability: 1
Header DbId: mdl
DbLabel: MEDLINE Ultimate
An: 38978399
AccessLevel: 2
PubType: Academic Journal
PubTypeId: academicJournal
PreciseRelevancyScore: 0
IllustrationInfo
Items – Name: Title
  Label: Title
  Group: Ti
  Data: Relevance of G protein-coupled receptor (GPCR) dynamics for receptor activation, signalling bias and allosteric modulation.
– Name: Author
  Label: Authors
  Group: Au
  Data: <searchLink fieldCode="AU" term="%22Lopez-Balastegui+M%22">Lopez-Balastegui M</searchLink>; Research Programme on Biomedical Informatics (GRIB), Hospital del Mar Medical Research Institute & Pompeu Fabra University, Barcelona, Spain.<br /><searchLink fieldCode="AU" term="%22Stepniewski+TM%22">Stepniewski TM</searchLink>; Research Programme on Biomedical Informatics (GRIB), Hospital del Mar Medical Research Institute & Pompeu Fabra University, Barcelona, Spain.; InterAx Biotech AG, Villigen, Switzerland.<br /><searchLink fieldCode="AU" term="%22Kogut-Günthel+MM%22">Kogut-Günthel MM</searchLink>; Leibniz Institute for Food Systems Biology at the Technical University of Munich, Freising, Germany.<br /><searchLink fieldCode="AU" term="%22Di+Pizio+A%22">Di Pizio A</searchLink>; Leibniz Institute for Food Systems Biology at the Technical University of Munich, Freising, Germany.; Chair for Chemoinformatics and Protein Modelling, Department of Molecular Life Science, School of Science, Technical University of Munich, Freising, Germany.<br /><searchLink fieldCode="AU" term="%22Rosenkilde+MM%22">Rosenkilde MM</searchLink>; Department of Biomedical Sciences, Faculty of Health and Medical Sciences University of Copenhagen, København N, Denmark.<br /><searchLink fieldCode="AU" term="%22Mao+J%22">Mao J</searchLink>; Huairou Research Center, Institute of Chemistry, Chinese Academy of Sciences, Beijing, China.<br /><searchLink fieldCode="AU" term="%22Selent+J%22">Selent J</searchLink>; Research Programme on Biomedical Informatics (GRIB), Hospital del Mar Medical Research Institute & Pompeu Fabra University, Barcelona, Spain.
– Name: TitleSource
  Label: Source
  Group: Src
  Data: <searchLink fieldCode="JN" term="%227502536%22">British journal of pharmacology</searchLink> [Br J Pharmacol] 2025 Jul; Vol. 182 (14), pp. 3211-3224. <i>Date of Electronic Publication: </i>2024 Jul 08.
– Name: TypePub
  Label: Publication Type
  Group: TypPub
  Data: Journal Article; Review
– Name: TitleSource
  Label: Journal Info
  Group: Src
  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Wiley%22">Wiley </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>7502536 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1476-5381 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200071188%22">00071188 </searchLink><i>NLM ISO Abbreviation: </i>Br J Pharmacol <i>Subsets: </i>MEDLINE
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=38978399
RecordInfo BibRecord:
  BibEntity:
    Identifiers:
      – Type: doi
        Value: 10.1111/bph.16495
    Languages:
      – Code: eng
        Text: English
    PhysicalDescription:
      Pagination:
        StartPage: 3211
    Titles:
      – TitleFull: Relevance of G protein-coupled receptor (GPCR) dynamics for receptor activation, signalling bias and allosteric modulation.
        Type: main
  BibRelationships:
    HasContributorRelationships:
      – PersonEntity:
          Name:
            NameFull: Lopez-Balastegui M
      – PersonEntity:
          Name:
            NameFull: Stepniewski TM
      – PersonEntity:
          Name:
            NameFull: Kogut-Günthel MM
      – PersonEntity:
          Name:
            NameFull: Di Pizio A
      – PersonEntity:
          Name:
            NameFull: Rosenkilde MM
      – PersonEntity:
          Name:
            NameFull: Mao J
      – PersonEntity:
          Name:
            NameFull: Selent J
    IsPartOfRelationships:
      – BibEntity:
          Dates:
            – D: 01
              M: 07
              Text: 2025 Jul
              Type: published
              Y: 2025
          Identifiers:
            – Type: issn-electronic
              Value: 1476-5381
          Numbering:
            – Type: volume
              Value: 182
            – Type: issue
              Value: 14
          Titles:
            – TitleFull: British journal of pharmacology
              Type: main
ResultId 1