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4-(3-Phenylsulfonylindol-2-yl)-1-(pyridin-2-yl)piperazinyl-methanones as Potent Inhibitors of both SARS-CoV-2 and HCoV-OC43 Viruses.

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Title: 4-(3-Phenylsulfonylindol-2-yl)-1-(pyridin-2-yl)piperazinyl-methanones as Potent Inhibitors of both SARS-CoV-2 and HCoV-OC43 Viruses.
Authors: Puxeddu M; Laboratory Affiliated to Istituto Pasteur Italia - Fondazione Cenci Bolognetti, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, I-00185 Rome, Italy., Donalisio M; Department of Clinical and Biological Sciences, University of Turin, Regione Gonzole 10, I-10043 Orbassano, Turin, Italy., Bugert JJ; Institut für Mikrobiologie der Bundeswehr, Neuherbergstrasse 11, D-80937 München, Germany., Corona A; Department of Life and Environmental Sciences, University of Cagliari, S.P. 8 Monserrato, Sestu Km 0.700, I-09042 Monserrato, Italy., Cocomazzi P; Biophysics Institute, CNR-IBF, Via Corti 12, I-20133 Milan, Italy., Milani M; Biophysics Institute, CNR-IBF, Via Corti 12, I-20133 Milan, Italy., Hucke F; Institut für Mikrobiologie der Bundeswehr, Neuherbergstrasse 11, D-80937 München, Germany., Arduino I; Department of Clinical and Biological Sciences, University of Turin, Regione Gonzole 10, I-10043 Orbassano, Turin, Italy., Esposito F; Department of Life and Environmental Sciences, University of Cagliari, S.P. 8 Monserrato, Sestu Km 0.700, I-09042 Monserrato, Italy., Moretti P; DISVA, Department of Life Sciences and Environment, Università Politecnica delle Marche, Via Brecce Bianche, I-60131 Ancona, Italy., Ortore MG; DISVA, Department of Life Sciences and Environment, Università Politecnica delle Marche, Via Brecce Bianche, I-60131 Ancona, Italy., Nalli M; Laboratory Affiliated to Istituto Pasteur Italia - Fondazione Cenci Bolognetti, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, I-00185 Rome, Italy., Manetto S; Laboratory Affiliated to Istituto Pasteur Italia - Fondazione Cenci Bolognetti, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, I-00185 Rome, Italy., Mazzoccanti G; Laboratory Affiliated to Istituto Pasteur Italia - Fondazione Cenci Bolognetti, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, I-00185 Rome, Italy., Bigogno C; Aphad SrL, Via della Resistenza 65, 20090 Buccinasco, Italy., Dondio G; Aphad SrL, Via della Resistenza 65, 20090 Buccinasco, Italy., Sciò P; Laboratory Affiliated to Istituto Pasteur Italia - Fondazione Cenci Bolognetti, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, I-00185 Rome, Italy., Coluccia A; Laboratory Affiliated to Istituto Pasteur Italia - Fondazione Cenci Bolognetti, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, I-00185 Rome, Italy., Fracella M; Laboratory of Virology, Department of Molecular Medicine, Sapienza University of Rome, 00185 Rome, Italy., Antonelli G; Laboratory of Virology, Department of Molecular Medicine, Sapienza University of Rome, 00185 Rome, Italy., Lembo D; Department of Clinical and Biological Sciences, University of Turin, Regione Gonzole 10, I-10043 Orbassano, Turin, Italy., Tramontano E; Department of Life and Environmental Sciences, University of Cagliari, S.P. 8 Monserrato, Sestu Km 0.700, I-09042 Monserrato, Italy., Silvestri R; Laboratory Affiliated to Istituto Pasteur Italia - Fondazione Cenci Bolognetti, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, I-00185 Rome, Italy., Mastrangelo E; Biophysics Institute, CNR-IBF, Via Corti 12, I-20133 Milan, Italy., La Regina G; Laboratory Affiliated to Istituto Pasteur Italia - Fondazione Cenci Bolognetti, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, I-00185 Rome, Italy.
Source: ACS infectious diseases [ACS Infect Dis] 2024 Sep 13; Vol. 10 (9), pp. 3158-3175. Date of Electronic Publication: 2024 Aug 03.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: ACS Publications Country of Publication: United States NLM ID: 101654580 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2373-8227 (Electronic) Linking ISSN: 23738227 NLM ISO Abbreviation: ACS Infect Dis Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: 4-(3-Phenylsulfonylindol-2-yl)-1-(pyridin-2-yl)piperazinyl-methanones as Potent Inhibitors of both SARS-CoV-2 and HCoV-OC43 Viruses.
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  Data: <searchLink fieldCode="AU" term="%22Puxeddu+M%22">Puxeddu M</searchLink>; Laboratory Affiliated to Istituto Pasteur Italia - Fondazione Cenci Bolognetti, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, I-00185 Rome, Italy.<br /><searchLink fieldCode="AU" term="%22Donalisio+M%22">Donalisio M</searchLink>; Department of Clinical and Biological Sciences, University of Turin, Regione Gonzole 10, I-10043 Orbassano, Turin, Italy.<br /><searchLink fieldCode="AU" term="%22Bugert+JJ%22">Bugert JJ</searchLink>; Institut für Mikrobiologie der Bundeswehr, Neuherbergstrasse 11, D-80937 München, Germany.<br /><searchLink fieldCode="AU" term="%22Corona+A%22">Corona A</searchLink>; Department of Life and Environmental Sciences, University of Cagliari, S.P. 8 Monserrato, Sestu Km 0.700, I-09042 Monserrato, Italy.<br /><searchLink fieldCode="AU" term="%22Cocomazzi+P%22">Cocomazzi P</searchLink>; Biophysics Institute, CNR-IBF, Via Corti 12, I-20133 Milan, Italy.<br /><searchLink fieldCode="AU" term="%22Milani+M%22">Milani M</searchLink>; Biophysics Institute, CNR-IBF, Via Corti 12, I-20133 Milan, Italy.<br /><searchLink fieldCode="AU" term="%22Hucke+F%22">Hucke F</searchLink>; Institut für Mikrobiologie der Bundeswehr, Neuherbergstrasse 11, D-80937 München, Germany.<br /><searchLink fieldCode="AU" term="%22Arduino+I%22">Arduino I</searchLink>; Department of Clinical and Biological Sciences, University of Turin, Regione Gonzole 10, I-10043 Orbassano, Turin, Italy.<br /><searchLink fieldCode="AU" term="%22Esposito+F%22">Esposito F</searchLink>; Department of Life and Environmental Sciences, University of Cagliari, S.P. 8 Monserrato, Sestu Km 0.700, I-09042 Monserrato, Italy.<br /><searchLink fieldCode="AU" term="%22Moretti+P%22">Moretti P</searchLink>; DISVA, Department of Life Sciences and Environment, Università Politecnica delle Marche, Via Brecce Bianche, I-60131 Ancona, Italy.<br /><searchLink fieldCode="AU" term="%22Ortore+MG%22">Ortore MG</searchLink>; DISVA, Department of Life Sciences and Environment, Università Politecnica delle Marche, Via Brecce Bianche, I-60131 Ancona, Italy.<br /><searchLink fieldCode="AU" term="%22Nalli+M%22">Nalli M</searchLink>; 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Laboratory Affiliated to Istituto Pasteur Italia - Fondazione Cenci Bolognetti, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, I-00185 Rome, Italy.<br /><searchLink fieldCode="AU" term="%22Coluccia+A%22">Coluccia A</searchLink>; Laboratory Affiliated to Istituto Pasteur Italia - Fondazione Cenci Bolognetti, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, I-00185 Rome, Italy.<br /><searchLink fieldCode="AU" term="%22Fracella+M%22">Fracella M</searchLink>; Laboratory of Virology, Department of Molecular Medicine, Sapienza University of Rome, 00185 Rome, Italy.<br /><searchLink fieldCode="AU" term="%22Antonelli+G%22">Antonelli G</searchLink>; Laboratory of Virology, Department of Molecular Medicine, Sapienza University of Rome, 00185 Rome, Italy.<br /><searchLink fieldCode="AU" term="%22Lembo+D%22">Lembo D</searchLink>; Department of Clinical and Biological Sciences, University of Turin, Regione Gonzole 10, I-10043 Orbassano, Turin, Italy.<br /><searchLink fieldCode="AU" term="%22Tramontano+E%22">Tramontano E</searchLink>; Department of Life and Environmental Sciences, University of Cagliari, S.P. 8 Monserrato, Sestu Km 0.700, I-09042 Monserrato, Italy.<br /><searchLink fieldCode="AU" term="%22Silvestri+R%22">Silvestri R</searchLink>; Laboratory Affiliated to Istituto Pasteur Italia - Fondazione Cenci Bolognetti, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, I-00185 Rome, Italy.<br /><searchLink fieldCode="AU" term="%22Mastrangelo+E%22">Mastrangelo E</searchLink>; Biophysics Institute, CNR-IBF, Via Corti 12, I-20133 Milan, Italy.<br /><searchLink fieldCode="AU" term="%22La+Regina+G%22">La Regina G</searchLink>; Laboratory Affiliated to Istituto Pasteur Italia - Fondazione Cenci Bolognetti, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, I-00185 Rome, Italy.
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