Emerging therapeutics: The imidazo[1,2-b]pyridazine scaffold as a novel drug candidate for eumycetoma, a neglected tropical disease.

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Title: Emerging therapeutics: The imidazo[1,2-b]pyridazine scaffold as a novel drug candidate for eumycetoma, a neglected tropical disease.
Authors: Elkheir LYM; The Mycetoma Research Center, University of Khartoum, Khartoum, Sudan; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Khartoum, Sudan; EA 7502 Synthèse et Isolement de Molécules Bioactives (SIMBA), University of Tours, France., Delaye PO; EA 7502 Synthèse et Isolement de Molécules Bioactives (SIMBA), University of Tours, France., Penichon M; EA 7502 Synthèse et Isolement de Molécules Bioactives (SIMBA), University of Tours, France., Eadie K; Department of Microbiology and Infectious Diseases, Erasmus Medical Center, University of Rotterdam, the Netherlands., Mohamed MA; Department of Pharmaceutical Chemistry, College of Pharmacy, Jouf University, KSA, Saudi Arabia., Besson P; UMR INSERM U1327 ISCHEMIA 'Membrane signalling and inflammation in reperfusion injuries', University of Tours, France., Chesnay A; UMR INSERM U 1100 Centre d'Etudes des Pathologies Respiratoires, University of Tours, France., Desoubeaux G; UMR INSERM U 1100 Centre d'Etudes des Pathologies Respiratoires, University of Tours, France., Roger S; UMR INSERM U1327 ISCHEMIA 'Membrane signalling and inflammation in reperfusion injuries', University of Tours, France., van de Sande WWJ; Department of Microbiology and Infectious Diseases, Erasmus Medical Center, University of Rotterdam, the Netherlands., Fahal AH; The Mycetoma Research Center, University of Khartoum, Khartoum, Sudan., Enguehard-Gueiffier C; EA 7502 Synthèse et Isolement de Molécules Bioactives (SIMBA), University of Tours, France. Electronic address: cecile.gueiffier@univ-tours.fr.
Source: European journal of medicinal chemistry [Eur J Med Chem] 2024 Nov 05; Vol. 277, pp. 116720. Date of Electronic Publication: 2024 Jul 26.
Publication Type: Journal Article
Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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