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Cerastecin Inhibition of the Lipooligosaccharide Transporter MsbA to Combat Acinetobacter baumannii: From Screening Impurity to In Vivo Efficacy.

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Title: Cerastecin Inhibition of the Lipooligosaccharide Transporter MsbA to Combat Acinetobacter baumannii: From Screening Impurity to In Vivo Efficacy.
Authors: Skudlarek JW; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Cooke AJ; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Mitchell HJ; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Babaoglu K; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Shaw AW; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Tong L; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Nomland AB; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Labroli M; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Sha D; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Mulhearn JJ; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Wu C; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Li SW; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Beshore DC; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Hughes JME; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Jouffroy M; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Wang H; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Balibar CJ; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Painter RE; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Shen P; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Lange HS; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Ishchenko A; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Chen YT; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Klein DJ; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Tracy RW; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Miller RR; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Cabalu TD; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Wu Z; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Leithead A; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Scapin G; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Hruza AW; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Dzhekieva L; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Bukhtiyarova M; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Homsher MF; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Xu M; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Bahnck-Teets C; Merck & Co., Inc., Rahway, New Jersey 07065, United States., McKenney D; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Buevich AV; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Liu J; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Zhang LK; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Meng T; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Kelly T; Merck & Co., Inc., Rahway, New Jersey 07065, United States., DiNunzio E; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Soisson S; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Cheng RKY; leadXpro AG, CH-5234 Villigen, Switzerland., Hennig M; leadXpro AG, CH-5234 Villigen, Switzerland., Raheem I; Merck & Co., Inc., Rahway, New Jersey 07065, United States., Walker SS; Merck & Co., Inc., Rahway, New Jersey 07065, United States.
Source: Journal of medicinal chemistry [J Med Chem] 2024 Sep 12; Vol. 67 (17), pp. 15620-15675. Date of Electronic Publication: 2024 Aug 22.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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