Structure-Activity Relationship of Oxacyclo- and Triazolo-Containing Respiratory Syncytial Virus Polymerase Inhibitors.

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Title: Structure-Activity Relationship of Oxacyclo- and Triazolo-Containing Respiratory Syncytial Virus Polymerase Inhibitors.
Authors: Tran MT; Janssen Pharmaceutica NV, 2340 Beerse, Belgium., Grosse S; Janssen Pharmaceutica NV, 2340 Beerse, Belgium., Carbajo RJ; Janssen Research and Development, Janssen-Cilag, S.A., C/Jarama 75, 45007 Toledo, Spain., Jacoby E; Janssen Pharmaceutica NV, 2340 Beerse, Belgium., Yin Y; Johnson & Johnson Innovative Medicine, Spring House, Pennsylvania, Pennsylvania 19477, United States., Yu X; Johnson & Johnson Innovative Medicine, Spring House, Pennsylvania, Pennsylvania 19477, United States., Martinez C; Janssen Pharmaceutica NV, 2340 Beerse, Belgium., Stoops B; Janssen Pharmaceutica NV, 2340 Beerse, Belgium., Cooymans L; Janssen Pharmaceutica NV, 2340 Beerse, Belgium., Hu L; Janssen Pharmaceutica NV, 2340 Beerse, Belgium., Lutter FH; Chemical Process R&D, Discovery Process Research, Janssen Pharmaceutica NV, 2340 Beerse, Belgium., Pieters S; Janssen Pharmaceutica NV, 2340 Beerse, Belgium., Tan E; Janssen Pharmaceutica NV, 2340 Beerse, Belgium., Alcázar J; Janssen Research and Development, Janssen-Cilag, S.A., C/Jarama 75, 45007 Toledo, Spain., Roymans D; Janssen Pharmaceutica NV, 2340 Beerse, Belgium., van Vlijmen H; Janssen Pharmaceutica NV, 2340 Beerse, Belgium., Rigaux P; Janssen Pharmaceutica NV, 2340 Beerse, Belgium., Sharma S; Johnson & Johnson Innovative Medicine, Spring House, Pennsylvania, Pennsylvania 19477, United States., Jonckers THM; Janssen Pharmaceutica NV, 2340 Beerse, Belgium.
Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2024 Aug 02; Vol. 15 (9), pp. 1549-1558. Date of Electronic Publication: 2024 Aug 02 (Print Publication: 2024).
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1948-5875
DOI:10.1021/acsmedchemlett.4c00272