Pharmacodynamics of the orexin type 1 (OX1) receptor in colon cancer cell models: A two-sided nature of antagonistic ligands resulting from partial dissociation of Gq.
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| Title: | Pharmacodynamics of the orexin type 1 (OX |
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| Authors: | Gratio V; INSERM UMR1149/Inflammation Research Center (CRI), Team 'From Inflammation to Cancer in Digestive diseases (INDiD)', DHU UNITY, Université Paris Cité, Paris, France.; INSERM UMR1149/Inflammation Research Center (CRI), Flow Cytometry Platform (CytoCRI), DHU UNITY, Université Paris Cité, Paris, France., Dragan P; Faculty of Chemistry, University of Warsaw, Warsaw, Poland., Garcia L; INSERM UMR1149/Inflammation Research Center (CRI), Team 'From Inflammation to Cancer in Digestive diseases (INDiD)', DHU UNITY, Université Paris Cité, Paris, France., Saveanu L; INSERM UMR1149/Inflammation Research Center (CRI), Team 'Antigen Presentation by Dendritic Cells to T cells (APreT)', DHU UNITY, Université Paris Cité, Paris, France., Nicole P; INSERM UMR1149/Inflammation Research Center (CRI), Team 'From Inflammation to Cancer in Digestive diseases (INDiD)', DHU UNITY, Université Paris Cité, Paris, France., Voisin T; INSERM UMR1149/Inflammation Research Center (CRI), Team 'From Inflammation to Cancer in Digestive diseases (INDiD)', DHU UNITY, Université Paris Cité, Paris, France., Latek D; Faculty of Chemistry, University of Warsaw, Warsaw, Poland., Couvineau A; INSERM UMR1149/Inflammation Research Center (CRI), Team 'From Inflammation to Cancer in Digestive diseases (INDiD)', DHU UNITY, Université Paris Cité, Paris, France. |
| Source: | British journal of pharmacology [Br J Pharmacol] 2025 Apr; Vol. 182 (7), pp. 1528-1545. Date of Electronic Publication: 2024 Dec 15. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Wiley Country of Publication: England NLM ID: 7502536 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1476-5381 (Electronic) Linking ISSN: 00071188 NLM ISO Abbreviation: Br J Pharmacol Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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| ISSN: | 1476-5381 |
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| DOI: | 10.1111/bph.17422 |