Pharmacodynamics of the orexin type 1 (OX1) receptor in colon cancer cell models: A two-sided nature of antagonistic ligands resulting from partial dissociation of Gq.

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Title: Pharmacodynamics of the orexin type 1 (OX1) receptor in colon cancer cell models: A two-sided nature of antagonistic ligands resulting from partial dissociation of Gq.
Authors: Gratio V; INSERM UMR1149/Inflammation Research Center (CRI), Team 'From Inflammation to Cancer in Digestive diseases (INDiD)', DHU UNITY, Université Paris Cité, Paris, France.; INSERM UMR1149/Inflammation Research Center (CRI), Flow Cytometry Platform (CytoCRI), DHU UNITY, Université Paris Cité, Paris, France., Dragan P; Faculty of Chemistry, University of Warsaw, Warsaw, Poland., Garcia L; INSERM UMR1149/Inflammation Research Center (CRI), Team 'From Inflammation to Cancer in Digestive diseases (INDiD)', DHU UNITY, Université Paris Cité, Paris, France., Saveanu L; INSERM UMR1149/Inflammation Research Center (CRI), Team 'Antigen Presentation by Dendritic Cells to T cells (APreT)', DHU UNITY, Université Paris Cité, Paris, France., Nicole P; INSERM UMR1149/Inflammation Research Center (CRI), Team 'From Inflammation to Cancer in Digestive diseases (INDiD)', DHU UNITY, Université Paris Cité, Paris, France., Voisin T; INSERM UMR1149/Inflammation Research Center (CRI), Team 'From Inflammation to Cancer in Digestive diseases (INDiD)', DHU UNITY, Université Paris Cité, Paris, France., Latek D; Faculty of Chemistry, University of Warsaw, Warsaw, Poland., Couvineau A; INSERM UMR1149/Inflammation Research Center (CRI), Team 'From Inflammation to Cancer in Digestive diseases (INDiD)', DHU UNITY, Université Paris Cité, Paris, France.
Source: British journal of pharmacology [Br J Pharmacol] 2025 Apr; Vol. 182 (7), pp. 1528-1545. Date of Electronic Publication: 2024 Dec 15.
Publication Type: Journal Article
Journal Info: Publisher: Wiley Country of Publication: England NLM ID: 7502536 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1476-5381 (Electronic) Linking ISSN: 00071188 NLM ISO Abbreviation: Br J Pharmacol Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:1476-5381
DOI:10.1111/bph.17422