Rational Design and Optimization of a Potent IDO1 Proteolysis Targeting Chimera (PROTAC).
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| Title: | Rational Design and Optimization of a Potent IDO1 Proteolysis Targeting Chimera (PROTAC). |
|---|---|
| Authors: | Monsen PJ, Bommi PV, Grigorescu AA, Lauing KL, Mao Y, Berardi P, Zhai L, Ojo O, Penco-Campillo M, Koch T, Egozi M, Jha SV, Dunne SF, Jiang H, Song G, Zhang F, Kregel S, Vaziri-Gohar A, Fanning S, Sanchez-Gomez P, Allen JM, Yamini B, Lukas RV, Wainwright DA, Schiltz GE |
| Source: | BioRxiv : the preprint server for biology [bioRxiv] 2025 Jan 08. Date of Electronic Publication: 2025 Jan 08. |
| Publication Type: | Journal Article; Preprint |
| Journal Info: | Country of Publication: United States NLM ID: 101680187 Publication Model: Electronic Cited Medium: Internet ISSN: 2692-8205 (Electronic) Linking ISSN: 26928205 NLM ISO Abbreviation: bioRxiv Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 39829781 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Rational Design and Optimization of a Potent IDO1 Proteolysis Targeting Chimera (PROTAC). – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Monsen+PJ%22">Monsen PJ</searchLink><br /><searchLink fieldCode="AU" term="%22Bommi+PV%22">Bommi PV</searchLink><br /><searchLink fieldCode="AU" term="%22Grigorescu+AA%22">Grigorescu AA</searchLink><br /><searchLink fieldCode="AU" term="%22Lauing+KL%22">Lauing KL</searchLink><br /><searchLink fieldCode="AU" term="%22Mao+Y%22">Mao Y</searchLink><br /><searchLink fieldCode="AU" term="%22Berardi+P%22">Berardi P</searchLink><br /><searchLink fieldCode="AU" term="%22Zhai+L%22">Zhai L</searchLink><br /><searchLink fieldCode="AU" term="%22Ojo+O%22">Ojo O</searchLink><br /><searchLink fieldCode="AU" term="%22Penco-Campillo+M%22">Penco-Campillo M</searchLink><br /><searchLink fieldCode="AU" term="%22Koch+T%22">Koch T</searchLink><br /><searchLink fieldCode="AU" term="%22Egozi+M%22">Egozi M</searchLink><br /><searchLink fieldCode="AU" term="%22Jha+SV%22">Jha SV</searchLink><br /><searchLink fieldCode="AU" term="%22Dunne+SF%22">Dunne SF</searchLink><br /><searchLink fieldCode="AU" term="%22Jiang+H%22">Jiang H</searchLink><br /><searchLink fieldCode="AU" term="%22Song+G%22">Song G</searchLink><br /><searchLink fieldCode="AU" term="%22Zhang+F%22">Zhang F</searchLink><br /><searchLink fieldCode="AU" term="%22Kregel+S%22">Kregel S</searchLink><br /><searchLink fieldCode="AU" term="%22Vaziri-Gohar+A%22">Vaziri-Gohar A</searchLink><br /><searchLink fieldCode="AU" term="%22Fanning+S%22">Fanning S</searchLink><br /><searchLink fieldCode="AU" term="%22Sanchez-Gomez+P%22">Sanchez-Gomez P</searchLink><br /><searchLink fieldCode="AU" term="%22Allen+JM%22">Allen JM</searchLink><br /><searchLink fieldCode="AU" term="%22Yamini+B%22">Yamini B</searchLink><br /><searchLink fieldCode="AU" term="%22Lukas+RV%22">Lukas RV</searchLink><br /><searchLink fieldCode="AU" term="%22Wainwright+DA%22">Wainwright DA</searchLink><br /><searchLink fieldCode="AU" term="%22Schiltz+GE%22">Schiltz GE</searchLink> – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101680187%22">BioRxiv : the preprint server for biology</searchLink> [bioRxiv] 2025 Jan 08. <i>Date of Electronic Publication: </i>2025 Jan 08. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article; Preprint – Name: TitleSource Label: Journal Info Group: Src Data: <i>Country of Publication: </i>United States <i>NLM ID: </i>101680187 <i>Publication Model: </i>Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>2692-8205 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2226928205%22">26928205 </searchLink><i>NLM ISO Abbreviation: </i>bioRxiv <i>Subsets: </i>PubMed not MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=39829781 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1101/2025.01.07.631731 Languages: – Code: eng Text: English Titles: – TitleFull: Rational Design and Optimization of a Potent IDO1 Proteolysis Targeting Chimera (PROTAC). Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Monsen PJ – PersonEntity: Name: NameFull: Bommi PV – PersonEntity: Name: NameFull: Grigorescu AA – PersonEntity: Name: NameFull: Lauing KL – PersonEntity: Name: NameFull: Mao Y – PersonEntity: Name: NameFull: Berardi P – PersonEntity: Name: NameFull: Zhai L – PersonEntity: Name: NameFull: Ojo O – PersonEntity: Name: NameFull: Penco-Campillo M – PersonEntity: Name: NameFull: Koch T – PersonEntity: Name: NameFull: Egozi M – PersonEntity: Name: NameFull: Jha SV – PersonEntity: Name: NameFull: Dunne SF – PersonEntity: Name: NameFull: Jiang H – PersonEntity: Name: NameFull: Song G – PersonEntity: Name: NameFull: Zhang F – PersonEntity: Name: NameFull: Kregel S – PersonEntity: Name: NameFull: Vaziri-Gohar A – PersonEntity: Name: NameFull: Fanning S – PersonEntity: Name: NameFull: Sanchez-Gomez P – PersonEntity: Name: NameFull: Allen JM – PersonEntity: Name: NameFull: Yamini B – PersonEntity: Name: NameFull: Lukas RV – PersonEntity: Name: NameFull: Wainwright DA – PersonEntity: Name: NameFull: Schiltz GE IsPartOfRelationships: – BibEntity: Dates: – D: 08 M: 01 Text: 2025 Jan 08 Type: published Y: 2025 Identifiers: – Type: issn-electronic Value: 2692-8205 Titles: – TitleFull: BioRxiv : the preprint server for biology Type: main |
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