Identifying a non-conserved site for achieving allosteric covalent inhibition of CECR2.
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| Title: | Identifying a non-conserved site for achieving allosteric covalent inhibition of CECR2. |
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| Authors: | Tang CL; School of Chinese Materia Medica, Nanjing University of Chinese Medicine, Nanjing, 210023, China.; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China., Li YQ; School of Chinese Materia Medica, Nanjing University of Chinese Medicine, Nanjing, 210023, China.; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China., Du XK; Center for Systems Biology, Department of Bioinformatics, School of Life Sciences, Suzhou Medical College of Soochow University, Suzhou, 215123, China., Fang XX; School of Chinese Materia Medica, Nanjing University of Chinese Medicine, Nanjing, 210023, China.; Zhongshan Institute for Drug Discovery, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Zhongshan, 528400, China., Guang YM; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China., Li PZ; School of Chinese Materia Medica, Nanjing University of Chinese Medicine, Nanjing, 210023, China.; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China., Chen S; School of Chinese Materia Medica, Nanjing University of Chinese Medicine, Nanjing, 210023, China.; Zhongshan Institute for Drug Discovery, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Zhongshan, 528400, China., Xue SY; School of Chinese Materia Medica, Nanjing University of Chinese Medicine, Nanjing, 210023, China.; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China., Yu JM; School of Chinese Materia Medica, Nanjing University of Chinese Medicine, Nanjing, 210023, China.; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China., Liu XY; Center for Systems Biology, Department of Bioinformatics, School of Life Sciences, Suzhou Medical College of Soochow University, Suzhou, 215123, China., Luo YP; Zhongshan Institute for Drug Discovery, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Zhongshan, 528400, China.; School of Pharmacy, Zunyi Medical University, Zunyi, 563000, China., Zhou LX; Zhongshan Institute for Drug Discovery, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Zhongshan, 528400, China.; School of Pharmacy, Guizhou Medical University, Guiyang, 550004, China., Luo C; School of Chinese Materia Medica, Nanjing University of Chinese Medicine, Nanjing, 210023, China.; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China.; Zhongshan Institute for Drug Discovery, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Zhongshan, 528400, China.; School of Pharmacy, Guizhou Medical University, Guiyang, 550004, China., Xiong H; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China. xionghuan@zidd.ac.cn.; Zhongshan Institute for Drug Discovery, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Zhongshan, 528400, China. xionghuan@zidd.ac.cn., Liang ZJ; Center for Systems Biology, Department of Bioinformatics, School of Life Sciences, Suzhou Medical College of Soochow University, Suzhou, 215123, China. zjliang@suda.edu.cn.; Jiangsu Province Engineering Research Center of Precision Diagnostics and Therapeutics Development, Soochow University, Suzhou, 215123, China. zjliang@suda.edu.cn., Ding H; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China. hding@simm.ac.cn.; School of Pharmacy, Guizhou Medical University, Guiyang, 550004, China. hding@simm.ac.cn. |
| Source: | Acta pharmacologica Sinica [Acta Pharmacol Sin] 2025 May; Vol. 46 (5), pp. 1476-1491. Date of Electronic Publication: 2025 Jan 20. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Nature Publishing Group Country of Publication: United States NLM ID: 100956087 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1745-7254 (Electronic) Linking ISSN: 16714083 NLM ISO Abbreviation: Acta Pharmacol Sin Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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