Evaluating reversible inhibitory drug-drug interactions: enzyme kinetics, and in vitro-to-in vivo scaling models.

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Title: Evaluating reversible inhibitory drug-drug interactions: enzyme kinetics, and in vitro-to-in vivo scaling models.
Authors: Zhang Q; Department of Pharmacotherapy and Translational Research, University of Florida, 1345 Center Drive, Gainesville, FL 32610, United States., Greenblatt DJ; Program in Pharmacology and Drug Development, Tufts University School of Medicine, 136 Harrison Ave, Boston, MA 02111, United States., Melchert PW; Department of Pharmacotherapy and Translational Research, University of Florida, 1345 Center Drive, Gainesville, FL 32610, United States., Markowitz JS; Department of Pharmacotherapy and Translational Research, University of Florida, 1345 Center Drive, Gainesville, FL 32610, United States.; Center for Pharmacogenomics and Precision Medicine, University of Florida, 1345 Center Drive, Gainesville, FL 32610, United States.
Source: The Journal of pharmacy and pharmacology [J Pharm Pharmacol] 2025 Aug 04; Vol. 77 (8), pp. 1002-1010.
Publication Type: Journal Article
Journal Info: Publisher: Oxford University Press Country of Publication: England NLM ID: 0376363 Publication Model: Print Cited Medium: Internet ISSN: 2042-7158 (Electronic) Linking ISSN: 00223573 NLM ISO Abbreviation: J Pharm Pharmacol Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: <searchLink fieldCode="AU" term="%22Zhang+Q%22">Zhang Q</searchLink>; Department of Pharmacotherapy and Translational Research, University of Florida, 1345 Center Drive, Gainesville, FL 32610, United States.<br /><searchLink fieldCode="AU" term="%22Greenblatt+DJ%22">Greenblatt DJ</searchLink>; Program in Pharmacology and Drug Development, Tufts University School of Medicine, 136 Harrison Ave, Boston, MA 02111, United States.<br /><searchLink fieldCode="AU" term="%22Melchert+PW%22">Melchert PW</searchLink>; Department of Pharmacotherapy and Translational Research, University of Florida, 1345 Center Drive, Gainesville, FL 32610, United States.<br /><searchLink fieldCode="AU" term="%22Markowitz+JS%22">Markowitz JS</searchLink>; Department of Pharmacotherapy and Translational Research, University of Florida, 1345 Center Drive, Gainesville, FL 32610, United States.; Center for Pharmacogenomics and Precision Medicine, University of Florida, 1345 Center Drive, Gainesville, FL 32610, United States.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Oxford+University+Press%22">Oxford University Press </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>0376363 <i>Publication Model: </i>Print <i>Cited Medium: </i>Internet <i>ISSN: </i>2042-7158 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200223573%22">00223573 </searchLink><i>NLM ISO Abbreviation: </i>J Pharm Pharmacol <i>Subsets: </i>MEDLINE
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        Value: 10.1093/jpp/rgaf029
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        Text: English
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              Text: 2025 Aug 04
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              Y: 2025
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