Investigation of an OATP1B inhibitory effect by a cyclic peptide using the endogenous biomarker coproporphyrin-I in monkeys.

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Title: Investigation of an OATP1B inhibitory effect by a cyclic peptide using the endogenous biomarker coproporphyrin-I in monkeys.
Authors: Sawada H; Laboratory for Drug Discovery and Development, Shionogi & Co., Ltd, Japan., Kido Y; Laboratory for Drug Discovery and Development, Shionogi & Co., Ltd, Japan., Iwasaki M; Department of Biological Material Generation, Shionogi TechnoAdvance Research & Co., Ltd, Japan., Nishida K; Corporate Planning Division, Shionogi TechnoAdvance Research & Co., Ltd, Japan., Mayumi K; Drug Development and Regulatory Science Division, Shionogi & Co., Ltd, Japan., Watari R; Laboratory for Drug Discovery and Development, Shionogi & Co., Ltd, Japan. Electronic address: ryosuke.watari@shionogi.co.jp.
Source: Drug metabolism and pharmacokinetics [Drug Metab Pharmacokinet] 2025 Aug; Vol. 63, pp. 101497. Date of Electronic Publication: 2025 Jun 03.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Country of Publication: England NLM ID: 101164773 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1880-0920 (Electronic) Linking ISSN: 13474367 NLM ISO Abbreviation: Drug Metab Pharmacokinet Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1880-0920
DOI:10.1016/j.dmpk.2025.101497