SAG1.3-derived Frizzled-targeting small-molecule compounds.

Saved in:
Bibliographic Details
Title: SAG1.3-derived Frizzled-targeting small-molecule compounds.
Authors: Grätz L; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden., Turku A; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden., Kozielewicz P; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden., Bowin CF; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden., Scharf MM; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden., Voss JH; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden., Kinsolving J; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden., Shekhani R; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden., Oliva-Vilarnau N; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Personalized Medicine and Drug Development, Biomedicum, Stockholm, Sweden., Koolmeister T; Chemical Biology Consortium Sweden, Science for Life Laboratory, Department of Medical Biochemistry and Biophysics, Karolinska Institutet, Stockholm, Sweden., Körber M; Department of Chemistry and Pharmacy, Friedrich-Alexander-Universität Erlangen-Nürnberg, Erlangen, Germany., Lauschke VM; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Personalized Medicine and Drug Development, Biomedicum, Stockholm, Sweden; Dr Margarete Fischer-Bosch Institute of Clinical Pharmacology, Translational Pharmacology and Drug Discovery, Stuttgart, Germany; University of Tübingen, Tübingen, Germany., Löber S; Department of Chemistry and Pharmacy, Friedrich-Alexander-Universität Erlangen-Nürnberg, Erlangen, Germany; FAUNeW - Research Center New Bioactive Compounds, Friedrich-Alexander-Universität Erlangen-Nürnberg, Erlangen, Germany., Gmeiner P; Department of Chemistry and Pharmacy, Friedrich-Alexander-Universität Erlangen-Nürnberg, Erlangen, Germany; FAUNeW - Research Center New Bioactive Compounds, Friedrich-Alexander-Universität Erlangen-Nürnberg, Erlangen, Germany., Schulte G; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden. Electronic address: gunnar.schulte@ki.se.
Source: The Journal of biological chemistry [J Biol Chem] 2025 Nov; Vol. 301 (11), pp. 110751. Date of Electronic Publication: 2025 Sep 22.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Elsevier Inc. on behalf of American Society for Biochemistry and Molecular Biology Country of Publication: United States NLM ID: 2985121R Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1083-351X (Electronic) Linking ISSN: 00219258 NLM ISO Abbreviation: J Biol Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
FullText Text:
  Availability: 0
Header DbId: mdl
DbLabel: MEDLINE Ultimate
An: 40992662
AccessLevel: 2
PubType: Academic Journal
PubTypeId: academicJournal
PreciseRelevancyScore: 0
IllustrationInfo
Items – Name: Title
  Label: Title
  Group: Ti
  Data: SAG1.3-derived Frizzled-targeting small-molecule compounds.
– Name: Author
  Label: Authors
  Group: Au
  Data: <searchLink fieldCode="AU" term="%22Grätz+L%22">Grätz L</searchLink>; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden.<br /><searchLink fieldCode="AU" term="%22Turku+A%22">Turku A</searchLink>; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden.<br /><searchLink fieldCode="AU" term="%22Kozielewicz+P%22">Kozielewicz P</searchLink>; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden.<br /><searchLink fieldCode="AU" term="%22Bowin+CF%22">Bowin CF</searchLink>; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden.<br /><searchLink fieldCode="AU" term="%22Scharf+MM%22">Scharf MM</searchLink>; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden.<br /><searchLink fieldCode="AU" term="%22Voss+JH%22">Voss JH</searchLink>; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden.<br /><searchLink fieldCode="AU" term="%22Kinsolving+J%22">Kinsolving J</searchLink>; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden.<br /><searchLink fieldCode="AU" term="%22Shekhani+R%22">Shekhani R</searchLink>; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden.<br /><searchLink fieldCode="AU" term="%22Oliva-Vilarnau+N%22">Oliva-Vilarnau N</searchLink>; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Personalized Medicine and Drug Development, Biomedicum, Stockholm, Sweden.<br /><searchLink fieldCode="AU" term="%22Koolmeister+T%22">Koolmeister T</searchLink>; Chemical Biology Consortium Sweden, Science for Life Laboratory, Department of Medical Biochemistry and Biophysics, Karolinska Institutet, Stockholm, Sweden.<br /><searchLink fieldCode="AU" term="%22Körber+M%22">Körber M</searchLink>; Department of Chemistry and Pharmacy, Friedrich-Alexander-Universität Erlangen-Nürnberg, Erlangen, Germany.<br /><searchLink fieldCode="AU" term="%22Lauschke+VM%22">Lauschke VM</searchLink>; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Personalized Medicine and Drug Development, Biomedicum, Stockholm, Sweden; Dr Margarete Fischer-Bosch Institute of Clinical Pharmacology, Translational Pharmacology and Drug Discovery, Stuttgart, Germany; University of Tübingen, Tübingen, Germany.<br /><searchLink fieldCode="AU" term="%22Löber+S%22">Löber S</searchLink>; Department of Chemistry and Pharmacy, Friedrich-Alexander-Universität Erlangen-Nürnberg, Erlangen, Germany; FAUNeW - Research Center New Bioactive Compounds, Friedrich-Alexander-Universität Erlangen-Nürnberg, Erlangen, Germany.<br /><searchLink fieldCode="AU" term="%22Gmeiner+P%22">Gmeiner P</searchLink>; Department of Chemistry and Pharmacy, Friedrich-Alexander-Universität Erlangen-Nürnberg, Erlangen, Germany; FAUNeW - Research Center New Bioactive Compounds, Friedrich-Alexander-Universität Erlangen-Nürnberg, Erlangen, Germany.<br /><searchLink fieldCode="AU" term="%22Schulte+G%22">Schulte G</searchLink>; Karolinska Institutet, Department Physiology & Pharmacology, Sec. Receptor Biology & Signaling, Biomedicum, Stockholm, Sweden. Electronic address: gunnar.schulte@ki.se.
– Name: TitleSource
  Label: Source
  Group: Src
  Data: <searchLink fieldCode="JN" term="%222985121R%22">The Journal of biological chemistry</searchLink> [J Biol Chem] 2025 Nov; Vol. 301 (11), pp. 110751. <i>Date of Electronic Publication: </i>2025 Sep 22.
– Name: TypePub
  Label: Publication Type
  Group: TypPub
  Data: Journal Article; Research Support, Non-U.S. Gov't
– Name: TitleSource
  Label: Journal Info
  Group: Src
  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Inc%2E+on+behalf+of+American+Society+for+Biochemistry+and+Molecular+Biology%22">Elsevier Inc. on behalf of American Society for Biochemistry and Molecular Biology </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>2985121R <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1083-351X (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200219258%22">00219258 </searchLink><i>NLM ISO Abbreviation: </i>J Biol Chem <i>Subsets: </i>MEDLINE
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=40992662
RecordInfo BibRecord:
  BibEntity:
    Identifiers:
      – Type: doi
        Value: 10.1016/j.jbc.2025.110751
    Languages:
      – Code: eng
        Text: English
    PhysicalDescription:
      Pagination:
        StartPage: 110751
    Titles:
      – TitleFull: SAG1.3-derived Frizzled-targeting small-molecule compounds.
        Type: main
  BibRelationships:
    HasContributorRelationships:
      – PersonEntity:
          Name:
            NameFull: Grätz L
      – PersonEntity:
          Name:
            NameFull: Turku A
      – PersonEntity:
          Name:
            NameFull: Kozielewicz P
      – PersonEntity:
          Name:
            NameFull: Bowin CF
      – PersonEntity:
          Name:
            NameFull: Scharf MM
      – PersonEntity:
          Name:
            NameFull: Voss JH
      – PersonEntity:
          Name:
            NameFull: Kinsolving J
      – PersonEntity:
          Name:
            NameFull: Shekhani R
      – PersonEntity:
          Name:
            NameFull: Oliva-Vilarnau N
      – PersonEntity:
          Name:
            NameFull: Koolmeister T
      – PersonEntity:
          Name:
            NameFull: Körber M
      – PersonEntity:
          Name:
            NameFull: Lauschke VM
      – PersonEntity:
          Name:
            NameFull: Löber S
      – PersonEntity:
          Name:
            NameFull: Gmeiner P
      – PersonEntity:
          Name:
            NameFull: Schulte G
    IsPartOfRelationships:
      – BibEntity:
          Dates:
            – D: 01
              M: 11
              Text: 2025 Nov
              Type: published
              Y: 2025
          Identifiers:
            – Type: issn-electronic
              Value: 1083-351X
          Numbering:
            – Type: volume
              Value: 301
            – Type: issue
              Value: 11
          Titles:
            – TitleFull: The Journal of biological chemistry
              Type: main
ResultId 1