Dual EZH1/2 inhibition enhances DNMT inhibitor efficacy in colon cancer through targeting H3K27me1.

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Title: Dual EZH1/2 inhibition enhances DNMT inhibitor efficacy in colon cancer through targeting H3K27me1.
Authors: Chomiak AA; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, USA., Wiseman AK; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, USA., Hrit J; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, USA., Liu Y; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, USA.; Van Andel Institute Graduate School, Grand Rapids, Michigan 49503, USA., Stransky S; Department of Biochemistry, Albert Einstein College of Medicine, Bronx, New York 10461, USA., Sidoli S; Department of Biochemistry, Albert Einstein College of Medicine, Bronx, New York 10461, USA., Tiedemann RL; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, USA., Rothbart SB; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, USA.; Van Andel Institute Graduate School, Grand Rapids, Michigan 49503, USA.
Source: BioRxiv : the preprint server for biology [bioRxiv] 2025 Sep 18. Date of Electronic Publication: 2025 Sep 18.
Publication Type: Journal Article; Preprint
Journal Info: Country of Publication: United States NLM ID: 101680187 Publication Model: Electronic Cited Medium: Internet ISSN: 2692-8205 (Electronic) Linking ISSN: 26928205 NLM ISO Abbreviation: bioRxiv Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
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PubType: Academic Journal
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  Data: Dual EZH1/2 inhibition enhances DNMT inhibitor efficacy in colon cancer through targeting H3K27me1.
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  Data: <searchLink fieldCode="AU" term="%22Chomiak+AA%22">Chomiak AA</searchLink>; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, USA.<br /><searchLink fieldCode="AU" term="%22Wiseman+AK%22">Wiseman AK</searchLink>; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, USA.<br /><searchLink fieldCode="AU" term="%22Hrit+J%22">Hrit J</searchLink>; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, USA.<br /><searchLink fieldCode="AU" term="%22Liu+Y%22">Liu Y</searchLink>; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, USA.; Van Andel Institute Graduate School, Grand Rapids, Michigan 49503, USA.<br /><searchLink fieldCode="AU" term="%22Stransky+S%22">Stransky S</searchLink>; Department of Biochemistry, Albert Einstein College of Medicine, Bronx, New York 10461, USA.<br /><searchLink fieldCode="AU" term="%22Sidoli+S%22">Sidoli S</searchLink>; Department of Biochemistry, Albert Einstein College of Medicine, Bronx, New York 10461, USA.<br /><searchLink fieldCode="AU" term="%22Tiedemann+RL%22">Tiedemann RL</searchLink>; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, USA.<br /><searchLink fieldCode="AU" term="%22Rothbart+SB%22">Rothbart SB</searchLink>; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, USA.; Van Andel Institute Graduate School, Grand Rapids, Michigan 49503, USA.
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  Data: <searchLink fieldCode="JN" term="%22101680187%22">BioRxiv : the preprint server for biology</searchLink> [bioRxiv] 2025 Sep 18. <i>Date of Electronic Publication: </i>2025 Sep 18.
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        Value: 10.1101/2025.09.16.676613
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              Text: 2025 Sep 18
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