Development of a Real-Time Fluorescence-Based Deamination Assay and Identification of Inhibitors of Human Cytidine Deaminase.

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Bibliographic Details
Title: Development of a Real-Time Fluorescence-Based Deamination Assay and Identification of Inhibitors of Human Cytidine Deaminase.
Authors: Moorthy R; Department of Medicinal Chemistry, University of Minnesota, Minneapolis, Minnesota 55455, United States., Grillo MJ; Department of Medicinal Chemistry, University of Minnesota, Minneapolis, Minnesota 55455, United States., Baur JW; Department of Chemistry, University of Minnesota, Minneapolis, Minnesota 55455, United States., Schmidt SA; Department of Chemistry, University of Minnesota, Minneapolis, Minnesota 55455, United States., Passow KT; Department of Medicinal Chemistry, University of Minnesota, Minneapolis, Minnesota 55455, United States., Demir Ö; Department of Molecular Biology, University of California - San Diego, La Jolla, California 92093, United States., Tang J; Department of Medicinal Chemistry, University of Minnesota, Minneapolis, Minnesota 55455, United States., Olson ME; Department of Medicinal Chemistry, University of Minnesota, Minneapolis, Minnesota 55455, United States., Amaro RE; Department of Molecular Biology, University of California - San Diego, La Jolla, California 92093, United States., Harki DA; Department of Medicinal Chemistry, University of Minnesota, Minneapolis, Minnesota 55455, United States.; Department of Chemistry, University of Minnesota, Minneapolis, Minnesota 55455, United States.
Source: ACS chemical biology [ACS Chem Biol] 2025 Nov 21; Vol. 20 (11), pp. 2593-2600. Date of Electronic Publication: 2025 Oct 22.
Publication Type: Journal Article; Research Support, N.I.H., Extramural
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101282906 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1554-8937 (Electronic) Linking ISSN: 15548929 NLM ISO Abbreviation: ACS Chem Biol Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1554-8937
DOI:10.1021/acschembio.5c00394