Toward the development of an innovative pharmacological compound employing peptides for EGFR-mediated drug delivery in anaplastic thyroid carcinoma.

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Title: Toward the development of an innovative pharmacological compound employing peptides for EGFR-mediated drug delivery in anaplastic thyroid carcinoma.
Authors: Kahvecioglu ZC; Unit of General, Organic and Biomedical Chemistry, NMR and Molecular Imaging Laboratory, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Avenue Victor Maistriau 19, Mendeleyev building, B-7000 Mons, Belgium. Electronic address: Zehracagla.KAHVECIOGLU@umons.ac.be., Vandecasteele S; Unit of General, Organic and Biomedical Chemistry, NMR and Molecular Imaging Laboratory, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Avenue Victor Maistriau 19, Mendeleyev building, B-7000 Mons, Belgium. Electronic address: samuel.vandecasteele@police.belgium.eu., Bougard M; Unit of General, Organic and Biomedical Chemistry, NMR and Molecular Imaging Laboratory, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Avenue Victor Maistriau 19, Mendeleyev building, B-7000 Mons, Belgium. Electronic address: Marine.Bougard@alumni.umons.ac.be., Rasson O; Unit of General, Organic and Biomedical Chemistry, NMR and Molecular Imaging Laboratory, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Avenue Victor Maistriau 19, Mendeleyev building, B-7000 Mons, Belgium. Electronic address: Olivia.Rasson@umons.ac.be., Nachtergael A; Unit of Therapeutic Chemistry and Pharmacognosy, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Chemin du Champ de Mars 25, B-7000 Mons, Belgium. Electronic address: Amandine.NACHTERGAEL@umons.ac.be., Duez P; Unit of Therapeutic Chemistry and Pharmacognosy, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Chemin du Champ de Mars 25, B-7000 Mons, Belgium. Electronic address: Pierre.DUEZ@umons.ac.be., Nonclercq D; Unit of Histology, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Pentagon building, Avenue du Champ de Mars 6, Pentagone building, B-7000 Mons, Belgium. Electronic address: Denis.NONCLERCQ@umons.ac.be., Remmelink M; Department of Pathological Anatomy, Erasme Hospital, Faculty of Medicine, Campus Erasme, CP 556, Route de Lennik, 808 1070 Bruxelles, Belgium. Electronic address: Myriam.Remmelink@hubruxelles.be., Laurent S; Unit of General, Organic and Biomedical Chemistry, NMR and Molecular Imaging Laboratory, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Avenue Victor Maistriau 19, Mendeleyev building, B-7000 Mons, Belgium; Center for Microscopy and Molecular Imaging (CMMI), rue Adrienne Bolland 8, B-6041 Gosselies, Belgium. Electronic address: Sophie.LAURENT@umons.ac.be., Saussez S; Human Anatomy and Experimental Oncology Unit, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Pentagon building, Avenue du Champ de Mars 6, B-7000 Mons, Belgium. Electronic address: Sven.SAUSSEZ@umosn.ac.be., Burtea C; Unit of General, Organic and Biomedical Chemistry, NMR and Molecular Imaging Laboratory, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Avenue Victor Maistriau 19, Mendeleyev building, B-7000 Mons, Belgium. Electronic address: Carmen.BURTEA@umons.ac.be.
Source: Biochemical pharmacology [Biochem Pharmacol] 2026 Jan; Vol. 243 (Pt 1), pp. 117448. Date of Electronic Publication: 2025 Oct 21.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Elsevier Science Country of Publication: England NLM ID: 0101032 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1873-2968 (Electronic) Linking ISSN: 00062952 NLM ISO Abbreviation: Biochem Pharmacol Subsets: MEDLINE
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  Data: Toward the development of an innovative pharmacological compound employing peptides for EGFR-mediated drug delivery in anaplastic thyroid carcinoma.
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  Data: <searchLink fieldCode="AU" term="%22Kahvecioglu+ZC%22">Kahvecioglu ZC</searchLink>; Unit of General, Organic and Biomedical Chemistry, NMR and Molecular Imaging Laboratory, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Avenue Victor Maistriau 19, Mendeleyev building, B-7000 Mons, Belgium. Electronic address: Zehracagla.KAHVECIOGLU@umons.ac.be.<br /><searchLink fieldCode="AU" term="%22Vandecasteele+S%22">Vandecasteele S</searchLink>; Unit of General, Organic and Biomedical Chemistry, NMR and Molecular Imaging Laboratory, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Avenue Victor Maistriau 19, Mendeleyev building, B-7000 Mons, Belgium. Electronic address: samuel.vandecasteele@police.belgium.eu.<br /><searchLink fieldCode="AU" term="%22Bougard+M%22">Bougard M</searchLink>; Unit of General, Organic and Biomedical Chemistry, NMR and Molecular Imaging Laboratory, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Avenue Victor Maistriau 19, Mendeleyev building, B-7000 Mons, Belgium. Electronic address: Marine.Bougard@alumni.umons.ac.be.<br /><searchLink fieldCode="AU" term="%22Rasson+O%22">Rasson O</searchLink>; Unit of General, Organic and Biomedical Chemistry, NMR and Molecular Imaging Laboratory, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Avenue Victor Maistriau 19, Mendeleyev building, B-7000 Mons, Belgium. Electronic address: Olivia.Rasson@umons.ac.be.<br /><searchLink fieldCode="AU" term="%22Nachtergael+A%22">Nachtergael A</searchLink>; Unit of Therapeutic Chemistry and Pharmacognosy, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Chemin du Champ de Mars 25, B-7000 Mons, Belgium. Electronic address: Amandine.NACHTERGAEL@umons.ac.be.<br /><searchLink fieldCode="AU" term="%22Duez+P%22">Duez P</searchLink>; Unit of Therapeutic Chemistry and Pharmacognosy, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Chemin du Champ de Mars 25, B-7000 Mons, Belgium. Electronic address: Pierre.DUEZ@umons.ac.be.<br /><searchLink fieldCode="AU" term="%22Nonclercq+D%22">Nonclercq D</searchLink>; Unit of Histology, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Pentagon building, Avenue du Champ de Mars 6, Pentagone building, B-7000 Mons, Belgium. Electronic address: Denis.NONCLERCQ@umons.ac.be.<br /><searchLink fieldCode="AU" term="%22Remmelink+M%22">Remmelink M</searchLink>; Department of Pathological Anatomy, Erasme Hospital, Faculty of Medicine, Campus Erasme, CP 556, Route de Lennik, 808 1070 Bruxelles, Belgium. Electronic address: Myriam.Remmelink@hubruxelles.be.<br /><searchLink fieldCode="AU" term="%22Laurent+S%22">Laurent S</searchLink>; Unit of General, Organic and Biomedical Chemistry, NMR and Molecular Imaging Laboratory, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Avenue Victor Maistriau 19, Mendeleyev building, B-7000 Mons, Belgium; Center for Microscopy and Molecular Imaging (CMMI), rue Adrienne Bolland 8, B-6041 Gosselies, Belgium. Electronic address: Sophie.LAURENT@umons.ac.be.<br /><searchLink fieldCode="AU" term="%22Saussez+S%22">Saussez S</searchLink>; Human Anatomy and Experimental Oncology Unit, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Pentagon building, Avenue du Champ de Mars 6, B-7000 Mons, Belgium. Electronic address: Sven.SAUSSEZ@umosn.ac.be.<br /><searchLink fieldCode="AU" term="%22Burtea+C%22">Burtea C</searchLink>; Unit of General, Organic and Biomedical Chemistry, NMR and Molecular Imaging Laboratory, Faculty of Medicine, Pharmacy and Biomedical Sciences, University of Mons, Avenue Victor Maistriau 19, Mendeleyev building, B-7000 Mons, Belgium. Electronic address: Carmen.BURTEA@umons.ac.be.
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  Data: <searchLink fieldCode="JN" term="%220101032%22">Biochemical pharmacology</searchLink> [Biochem Pharmacol] 2026 Jan; Vol. 243 (Pt 1), pp. 117448. <i>Date of Electronic Publication: </i>2025 Oct 21.
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        Value: 10.1016/j.bcp.2025.117448
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