Structure-guided allosteric modulation of the delta opioid receptor.

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Title: Structure-guided allosteric modulation of the delta opioid receptor.
Authors: Mobbs JI; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Parkville, Australia.; These authors contributed equally: Jesse I. Mobbs, M. Deborah Nguyen, Owindeep Deo., Nguyen MD; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.; These authors contributed equally: Jesse I. Mobbs, M. Deborah Nguyen, Owindeep Deo., Deo O; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.; These authors contributed equally: Jesse I. Mobbs, M. Deborah Nguyen, Owindeep Deo., Bartuzi D; Science for Life Laboratory, Department of Cell and Molecular Biology, Uppsala University, Uppsala, Sweden.; Department of Synthesis and Chemical Technology of Pharmaceutical Substances with Computer Modeling Laboratory, Faculty of Pharmacy, Medical University of Lublin, 4A Chodźki St., Lublin 20093, Poland., Venugopal H; Ramaciotti Centre for Cryo-Electron Microscopy, Monash University, Australia., Alvi S; Monash Institute of Pharmaceutical Sciences, Parkville, Australia., Pham V; Monash Institute of Pharmaceutical Sciences, Parkville, Australia., Barnes N; Monash Institute of Pharmaceutical Sciences, Parkville, Australia., Christopoulos A; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Parkville, Australia., Poole DP; Monash Institute of Pharmaceutical Sciences, Parkville, Australia., Carbone SE; Monash Institute of Pharmaceutical Sciences, Parkville, Australia., Jörg M; Monash Institute of Pharmaceutical Sciences, Parkville, Australia., Capuano B; Monash Institute of Pharmaceutical Sciences, Parkville, Australia., Carlsson J; Science for Life Laboratory, Department of Cell and Molecular Biology, Uppsala University, Uppsala, Sweden., Gondin AB; Monash Institute of Pharmaceutical Sciences, Parkville, Australia., Scammells PJ; Monash Institute of Pharmaceutical Sciences, Parkville, Australia., Valant C; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Parkville, Australia., Thal DM; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Parkville, Australia.
Source: BioRxiv : the preprint server for biology [bioRxiv] 2025 Oct 17. Date of Electronic Publication: 2025 Oct 17.
Publication Type: Journal Article; Preprint
Journal Info: Country of Publication: United States NLM ID: 101680187 Publication Model: Electronic Cited Medium: Internet ISSN: 2692-8205 (Electronic) Linking ISSN: 26928205 NLM ISO Abbreviation: bioRxiv Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
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  Data: Structure-guided allosteric modulation of the delta opioid receptor.
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  Data: <searchLink fieldCode="AU" term="%22Mobbs+JI%22">Mobbs JI</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Parkville, Australia.; These authors contributed equally: Jesse I. Mobbs, M. Deborah Nguyen, Owindeep Deo.<br /><searchLink fieldCode="AU" term="%22Nguyen+MD%22">Nguyen MD</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.; These authors contributed equally: Jesse I. Mobbs, M. Deborah Nguyen, Owindeep Deo.<br /><searchLink fieldCode="AU" term="%22Deo+O%22">Deo O</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.; These authors contributed equally: Jesse I. Mobbs, M. Deborah Nguyen, Owindeep Deo.<br /><searchLink fieldCode="AU" term="%22Bartuzi+D%22">Bartuzi D</searchLink>; Science for Life Laboratory, Department of Cell and Molecular Biology, Uppsala University, Uppsala, Sweden.; Department of Synthesis and Chemical Technology of Pharmaceutical Substances with Computer Modeling Laboratory, Faculty of Pharmacy, Medical University of Lublin, 4A Chodźki St., Lublin 20093, Poland.<br /><searchLink fieldCode="AU" term="%22Venugopal+H%22">Venugopal H</searchLink>; Ramaciotti Centre for Cryo-Electron Microscopy, Monash University, Australia.<br /><searchLink fieldCode="AU" term="%22Alvi+S%22">Alvi S</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.<br /><searchLink fieldCode="AU" term="%22Pham+V%22">Pham V</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.<br /><searchLink fieldCode="AU" term="%22Barnes+N%22">Barnes N</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.<br /><searchLink fieldCode="AU" term="%22Christopoulos+A%22">Christopoulos A</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Parkville, Australia.<br /><searchLink fieldCode="AU" term="%22Poole+DP%22">Poole DP</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.<br /><searchLink fieldCode="AU" term="%22Carbone+SE%22">Carbone SE</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.<br /><searchLink fieldCode="AU" term="%22Jörg+M%22">Jörg M</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.<br /><searchLink fieldCode="AU" term="%22Capuano+B%22">Capuano B</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.<br /><searchLink fieldCode="AU" term="%22Carlsson+J%22">Carlsson J</searchLink>; Science for Life Laboratory, Department of Cell and Molecular Biology, Uppsala University, Uppsala, Sweden.<br /><searchLink fieldCode="AU" term="%22Gondin+AB%22">Gondin AB</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.<br /><searchLink fieldCode="AU" term="%22Scammells+PJ%22">Scammells PJ</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.<br /><searchLink fieldCode="AU" term="%22Valant+C%22">Valant C</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Parkville, Australia.<br /><searchLink fieldCode="AU" term="%22Thal+DM%22">Thal DM</searchLink>; Monash Institute of Pharmaceutical Sciences, Parkville, Australia.; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Parkville, Australia.
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