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Biological Activity and Structural Biology of Current KAT6A Inhibitor Chemotypes.

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Title: Biological Activity and Structural Biology of Current KAT6A Inhibitor Chemotypes.
Authors: Suwandi A; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), Parkville, VIC 3052, Australia., Jin J; Institute for Advanced and Applied Chemical Synthesis, College of Pharmacy, Jinan University, Guangzhou, Guangdong 510632, China., Zhao Y; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), Parkville, VIC 3052, Australia., Mudududdla R; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), Parkville, VIC 3052, Australia., Gee YS; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), Parkville, VIC 3052, Australia., Deora GS; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), Parkville, VIC 3052, Australia., Sun Y; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), Parkville, VIC 3052, Australia., Wei H; School of Pharmaceutical Sciences, Nanjing Tech University, No. 30 South Puzhu Road, Nanjing 211816, People's Republic of China., Huang F; School of Pharmaceutical Sciences, Nanjing Tech University, No. 30 South Puzhu Road, Nanjing 211816, People's Republic of China., He JS; John Curtin School of Medical Research, Australian National University, Canberra, ACT 2600, Australia., George AJ; John Curtin School of Medical Research, Australian National University, Canberra, ACT 2600, Australia., Hermans SJ; ACRF Rational Drug Discovery Centre, St. Vincent's Institute of Medical Research, Fitzroy, VIC 3065, Australia.; Department of Biochemistry and Pharmacology, Bio21 Molecular Science and Biotechnology Institute, University of Melbourne, Melbourne, VIC 3010, Australia., Leaver DJ; School of Dentistry and Medical Sciences, Charles Sturt University, Wagga Wagga, NSW 2678, Australia., Parker MW; ACRF Rational Drug Discovery Centre, St. Vincent's Institute of Medical Research, Fitzroy, VIC 3065, Australia.; Department of Biochemistry and Pharmacology, Bio21 Molecular Science and Biotechnology Institute, University of Melbourne, Melbourne, VIC 3010, Australia., Baell JB; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), Parkville, VIC 3052, Australia.; School of Pharmaceutical Sciences, Nanjing Tech University, No. 30 South Puzhu Road, Nanjing 211816, People's Republic of China.; Australian Translational Medicinal Chemistry Facility (ATMCF), Monash University, Parkville, VIC 3052, Australia.
Source: Journal of medicinal chemistry [J Med Chem] 2026 Feb 12; Vol. 69 (3), pp. 2082-2114. Date of Electronic Publication: 2026 Jan 29.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Biological Activity and Structural Biology of Current KAT6A Inhibitor Chemotypes.
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  Data: <searchLink fieldCode="AU" term="%22Suwandi+A%22">Suwandi A</searchLink>; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), Parkville, VIC 3052, Australia.<br /><searchLink fieldCode="AU" term="%22Jin+J%22">Jin J</searchLink>; Institute for Advanced and Applied Chemical Synthesis, College of Pharmacy, Jinan University, Guangzhou, Guangdong 510632, China.<br /><searchLink fieldCode="AU" term="%22Zhao+Y%22">Zhao Y</searchLink>; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), Parkville, VIC 3052, Australia.<br /><searchLink fieldCode="AU" term="%22Mudududdla+R%22">Mudududdla R</searchLink>; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), Parkville, VIC 3052, Australia.<br /><searchLink fieldCode="AU" term="%22Gee+YS%22">Gee YS</searchLink>; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), Parkville, VIC 3052, Australia.<br /><searchLink fieldCode="AU" term="%22Deora+GS%22">Deora GS</searchLink>; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), Parkville, VIC 3052, Australia.<br /><searchLink fieldCode="AU" term="%22Sun+Y%22">Sun Y</searchLink>; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), Parkville, VIC 3052, Australia.<br /><searchLink fieldCode="AU" term="%22Wei+H%22">Wei H</searchLink>; School of Pharmaceutical Sciences, Nanjing Tech University, No. 30 South Puzhu Road, Nanjing 211816, People's Republic of China.<br /><searchLink fieldCode="AU" term="%22Huang+F%22">Huang F</searchLink>; School of Pharmaceutical Sciences, Nanjing Tech University, No. 30 South Puzhu Road, Nanjing 211816, People's Republic of China.<br /><searchLink fieldCode="AU" term="%22He+JS%22">He JS</searchLink>; John Curtin School of Medical Research, Australian National University, Canberra, ACT 2600, Australia.<br /><searchLink fieldCode="AU" term="%22George+AJ%22">George AJ</searchLink>; John Curtin School of Medical Research, Australian National University, Canberra, ACT 2600, Australia.<br /><searchLink fieldCode="AU" term="%22Hermans+SJ%22">Hermans SJ</searchLink>; ACRF Rational Drug Discovery Centre, St. Vincent's Institute of Medical Research, Fitzroy, VIC 3065, Australia.; Department of Biochemistry and Pharmacology, Bio21 Molecular Science and Biotechnology Institute, University of Melbourne, Melbourne, VIC 3010, Australia.<br /><searchLink fieldCode="AU" term="%22Leaver+DJ%22">Leaver DJ</searchLink>; School of Dentistry and Medical Sciences, Charles Sturt University, Wagga Wagga, NSW 2678, Australia.<br /><searchLink fieldCode="AU" term="%22Parker+MW%22">Parker MW</searchLink>; ACRF Rational Drug Discovery Centre, St. Vincent's Institute of Medical Research, Fitzroy, VIC 3065, Australia.; Department of Biochemistry and Pharmacology, Bio21 Molecular Science and Biotechnology Institute, University of Melbourne, Melbourne, VIC 3010, Australia.<br /><searchLink fieldCode="AU" term="%22Baell+JB%22">Baell JB</searchLink>; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University (Parkville Campus), Parkville, VIC 3052, Australia.; School of Pharmaceutical Sciences, Nanjing Tech University, No. 30 South Puzhu Road, Nanjing 211816, People's Republic of China.; Australian Translational Medicinal Chemistry Facility (ATMCF), Monash University, Parkville, VIC 3052, Australia.
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  Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 2026 Feb 12; Vol. 69 (3), pp. 2082-2114. <i>Date of Electronic Publication: </i>2026 Jan 29.
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        Value: 10.1021/acs.jmedchem.5c01426
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