Allosteric Induction of Estrogen Receptor Ligand Binding Domain Tetramerization by a Distinct Complete Estrogen Receptor Antagonist.

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Bibliographic Details
Title: Allosteric Induction of Estrogen Receptor Ligand Binding Domain Tetramerization by a Distinct Complete Estrogen Receptor Antagonist.
Authors: Fink EC; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States., Chawla R; Olema Oncology, San Francisco, California 94103, United States., Hancock GR; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States., Wells KS; Olema Oncology, San Francisco, California 94103, United States., Barratt S; Olema Oncology, San Francisco, California 94103, United States., Myles DC; Olema Oncology, San Francisco, California 94103, United States., Peña G; Olema Oncology, San Francisco, California 94103, United States., Robello BW; Olema Oncology, San Francisco, California 94103, United States., Hearn BR; Olema Oncology, San Francisco, California 94103, United States., Fanning SW; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States.
Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2026 Jan 16; Vol. 17 (2), pp. 441-449. Date of Electronic Publication: 2026 Jan 16 (Print Publication: 2026).
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1948-5875
DOI:10.1021/acsmedchemlett.5c00667