Allosteric Induction of Estrogen Receptor Ligand Binding Domain Tetramerization by a Distinct Complete Estrogen Receptor Antagonist.

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Title: Allosteric Induction of Estrogen Receptor Ligand Binding Domain Tetramerization by a Distinct Complete Estrogen Receptor Antagonist.
Authors: Fink EC; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States., Chawla R; Olema Oncology, San Francisco, California 94103, United States., Hancock GR; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States., Wells KS; Olema Oncology, San Francisco, California 94103, United States., Barratt S; Olema Oncology, San Francisco, California 94103, United States., Myles DC; Olema Oncology, San Francisco, California 94103, United States., Peña G; Olema Oncology, San Francisco, California 94103, United States., Robello BW; Olema Oncology, San Francisco, California 94103, United States., Hearn BR; Olema Oncology, San Francisco, California 94103, United States., Fanning SW; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States.
Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2026 Jan 16; Vol. 17 (2), pp. 441-449. Date of Electronic Publication: 2026 Jan 16 (Print Publication: 2026).
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE
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  Data: Allosteric Induction of Estrogen Receptor Ligand Binding Domain Tetramerization by a Distinct Complete Estrogen Receptor Antagonist.
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  Data: <searchLink fieldCode="AU" term="%22Fink+EC%22">Fink EC</searchLink>; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States.<br /><searchLink fieldCode="AU" term="%22Chawla+R%22">Chawla R</searchLink>; Olema Oncology, San Francisco, California 94103, United States.<br /><searchLink fieldCode="AU" term="%22Hancock+GR%22">Hancock GR</searchLink>; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States.<br /><searchLink fieldCode="AU" term="%22Wells+KS%22">Wells KS</searchLink>; Olema Oncology, San Francisco, California 94103, United States.<br /><searchLink fieldCode="AU" term="%22Barratt+S%22">Barratt S</searchLink>; Olema Oncology, San Francisco, California 94103, United States.<br /><searchLink fieldCode="AU" term="%22Myles+DC%22">Myles DC</searchLink>; Olema Oncology, San Francisco, California 94103, United States.<br /><searchLink fieldCode="AU" term="%22Peña+G%22">Peña G</searchLink>; Olema Oncology, San Francisco, California 94103, United States.<br /><searchLink fieldCode="AU" term="%22Robello+BW%22">Robello BW</searchLink>; Olema Oncology, San Francisco, California 94103, United States.<br /><searchLink fieldCode="AU" term="%22Hearn+BR%22">Hearn BR</searchLink>; Olema Oncology, San Francisco, California 94103, United States.<br /><searchLink fieldCode="AU" term="%22Fanning+SW%22">Fanning SW</searchLink>; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101521073 <i>Publication Model: </i>eCollection <i>Cited Medium: </i>Print <i>ISSN: </i>1948-5875 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2219485875%22">19485875 </searchLink><i>NLM ISO Abbreviation: </i>ACS Med Chem Lett <i>Subsets: </i>PubMed not MEDLINE
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        Value: 10.1021/acsmedchemlett.5c00667
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      – TitleFull: Allosteric Induction of Estrogen Receptor Ligand Binding Domain Tetramerization by a Distinct Complete Estrogen Receptor Antagonist.
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              Text: 2026 Jan 16
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