Allosteric Induction of Estrogen Receptor Ligand Binding Domain Tetramerization by a Distinct Complete Estrogen Receptor Antagonist.
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| Title: | Allosteric Induction of Estrogen Receptor Ligand Binding Domain Tetramerization by a Distinct Complete Estrogen Receptor Antagonist. |
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| Authors: | Fink EC; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States., Chawla R; Olema Oncology, San Francisco, California 94103, United States., Hancock GR; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States., Wells KS; Olema Oncology, San Francisco, California 94103, United States., Barratt S; Olema Oncology, San Francisco, California 94103, United States., Myles DC; Olema Oncology, San Francisco, California 94103, United States., Peña G; Olema Oncology, San Francisco, California 94103, United States., Robello BW; Olema Oncology, San Francisco, California 94103, United States., Hearn BR; Olema Oncology, San Francisco, California 94103, United States., Fanning SW; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States. |
| Source: | ACS medicinal chemistry letters [ACS Med Chem Lett] 2026 Jan 16; Vol. 17 (2), pp. 441-449. Date of Electronic Publication: 2026 Jan 16 (Print Publication: 2026). |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 41704390 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Allosteric Induction of Estrogen Receptor Ligand Binding Domain Tetramerization by a Distinct Complete Estrogen Receptor Antagonist. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Fink+EC%22">Fink EC</searchLink>; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States.<br /><searchLink fieldCode="AU" term="%22Chawla+R%22">Chawla R</searchLink>; Olema Oncology, San Francisco, California 94103, United States.<br /><searchLink fieldCode="AU" term="%22Hancock+GR%22">Hancock GR</searchLink>; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States.<br /><searchLink fieldCode="AU" term="%22Wells+KS%22">Wells KS</searchLink>; Olema Oncology, San Francisco, California 94103, United States.<br /><searchLink fieldCode="AU" term="%22Barratt+S%22">Barratt S</searchLink>; Olema Oncology, San Francisco, California 94103, United States.<br /><searchLink fieldCode="AU" term="%22Myles+DC%22">Myles DC</searchLink>; Olema Oncology, San Francisco, California 94103, United States.<br /><searchLink fieldCode="AU" term="%22Peña+G%22">Peña G</searchLink>; Olema Oncology, San Francisco, California 94103, United States.<br /><searchLink fieldCode="AU" term="%22Robello+BW%22">Robello BW</searchLink>; Olema Oncology, San Francisco, California 94103, United States.<br /><searchLink fieldCode="AU" term="%22Hearn+BR%22">Hearn BR</searchLink>; Olema Oncology, San Francisco, California 94103, United States.<br /><searchLink fieldCode="AU" term="%22Fanning+SW%22">Fanning SW</searchLink>; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101521073%22">ACS medicinal chemistry letters</searchLink> [ACS Med Chem Lett] 2026 Jan 16; Vol. 17 (2), pp. 441-449. <i>Date of Electronic Publication: </i>2026 Jan 16 (<i>Print Publication: </i>2026). – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101521073 <i>Publication Model: </i>eCollection <i>Cited Medium: </i>Print <i>ISSN: </i>1948-5875 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2219485875%22">19485875 </searchLink><i>NLM ISO Abbreviation: </i>ACS Med Chem Lett <i>Subsets: </i>PubMed not MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=41704390 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/acsmedchemlett.5c00667 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 441 Titles: – TitleFull: Allosteric Induction of Estrogen Receptor Ligand Binding Domain Tetramerization by a Distinct Complete Estrogen Receptor Antagonist. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Fink EC – PersonEntity: Name: NameFull: Chawla R – PersonEntity: Name: NameFull: Hancock GR – PersonEntity: Name: NameFull: Wells KS – PersonEntity: Name: NameFull: Barratt S – PersonEntity: Name: NameFull: Myles DC – PersonEntity: Name: NameFull: Peña G – PersonEntity: Name: NameFull: Robello BW – PersonEntity: Name: NameFull: Hearn BR – PersonEntity: Name: NameFull: Fanning SW IsPartOfRelationships: – BibEntity: Dates: – D: 16 M: 01 Text: 2026 Jan 16 Type: published Y: 2026 Identifiers: – Type: issn-print Value: 1948-5875 Numbering: – Type: volume Value: 17 – Type: issue Value: 2 Titles: – TitleFull: ACS medicinal chemistry letters Type: main |
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