Allosteric Induction of Estrogen Receptor Ligand Binding Domain Tetramerization by a Distinct Complete Estrogen Receptor Antagonist.
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| Title: | Allosteric Induction of Estrogen Receptor Ligand Binding Domain Tetramerization by a Distinct Complete Estrogen Receptor Antagonist. |
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| Authors: | Fink EC; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States., Chawla R; Olema Oncology, San Francisco, California 94103, United States., Hancock GR; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States., Wells KS; Olema Oncology, San Francisco, California 94103, United States., Barratt S; Olema Oncology, San Francisco, California 94103, United States., Myles DC; Olema Oncology, San Francisco, California 94103, United States., Peña G; Olema Oncology, San Francisco, California 94103, United States., Robello BW; Olema Oncology, San Francisco, California 94103, United States., Hearn BR; Olema Oncology, San Francisco, California 94103, United States., Fanning SW; Department of Cancer Biology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60546, United States. |
| Source: | ACS medicinal chemistry letters [ACS Med Chem Lett] 2026 Jan 16; Vol. 17 (2), pp. 441-449. Date of Electronic Publication: 2026 Jan 16 (Print Publication: 2026). |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
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