Quinoline carboxylic acid derivatives as potent ectonucleotidase inhibitors.

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Title: Quinoline carboxylic acid derivatives as potent ectonucleotidase inhibitors.
Authors: Ishaq A; Centre for Advanced Drug Research, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, 22060, Pakistan.; Department of Chemistry, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, 22060, Pakistan., Nawaz I; Centre for Advanced Drug Research, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, 22060, Pakistan., Qadir J; Centre for Advanced Drug Research, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, 22060, Pakistan., Alrokayan S; Research Chair for Biomedical Application of Nanomaterials, Biochemistry Department, College of Science, King Saud University, 11451, Riyadh, Saudi Arabia., Hussain T; Center of Excellence in Biotechnology Research, King Saud University, 11451, Riyadh, Saudi Arabia., Gelsleichter NE; Département de microbiologie-infectiologiee et d'immunologie, Centres PROTEO et ARThrite, Faculté de Médecine, Université Laval, Quebec City, QC, G1V 0A6, Canada.; Axe Maladies infectieuses et immunitaires, Centre de recherche du CHU de Québec, Université Laval, Quebec City, QC, G1V 4G2, Canada., Pelletier J; Axe Maladies infectieuses et immunitaires, Centre de recherche du CHU de Québec, Université Laval, Quebec City, QC, G1V 4G2, Canada., Sévigny J; Département de microbiologie-infectiologiee et d'immunologie, Centres PROTEO et ARThrite, Faculté de Médecine, Université Laval, Quebec City, QC, G1V 0A6, Canada.; Axe Maladies infectieuses et immunitaires, Centre de recherche du CHU de Québec, Université Laval, Quebec City, QC, G1V 4G2, Canada., Muhammad M; CAS Key Laboratory of Ion-Beam Bioengineering, Institute of Intelligent Machines, Hefei Institutes of Physical Science, Chinese Academy of Sciences, Hefei, China., Huang Q; CAS Key Laboratory of Ion-Beam Bioengineering, Institute of Intelligent Machines, Hefei Institutes of Physical Science, Chinese Academy of Sciences, Hefei, China.; Science Island Branch of Graduate School, University of Science and Technology of China, Hefei, China., Iqbal J; Centre for Advanced Drug Research, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, 22060, Pakistan. drjamshed@cuiatd.edu.pk.; Department of Chemistry, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, 22060, Pakistan. drjamshed@cuiatd.edu.pk.
Source: Scientific reports [Sci Rep] 2026 Feb 21; Vol. 16 (1). Date of Electronic Publication: 2026 Feb 21.
Publication Type: Journal Article
Journal Info: Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101563288 Publication Model: Electronic Cited Medium: Internet ISSN: 2045-2322 (Electronic) Linking ISSN: 20452322 NLM ISO Abbreviation: Sci Rep Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Quinoline carboxylic acid derivatives as potent ectonucleotidase inhibitors.
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  Data: <searchLink fieldCode="AU" term="%22Ishaq+A%22">Ishaq A</searchLink>; Centre for Advanced Drug Research, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, 22060, Pakistan.; Department of Chemistry, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, 22060, Pakistan.<br /><searchLink fieldCode="AU" term="%22Nawaz+I%22">Nawaz I</searchLink>; Centre for Advanced Drug Research, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, 22060, Pakistan.<br /><searchLink fieldCode="AU" term="%22Qadir+J%22">Qadir J</searchLink>; Centre for Advanced Drug Research, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, 22060, Pakistan.<br /><searchLink fieldCode="AU" term="%22Alrokayan+S%22">Alrokayan S</searchLink>; Research Chair for Biomedical Application of Nanomaterials, Biochemistry Department, College of Science, King Saud University, 11451, Riyadh, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Hussain+T%22">Hussain T</searchLink>; Center of Excellence in Biotechnology Research, King Saud University, 11451, Riyadh, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Gelsleichter+NE%22">Gelsleichter NE</searchLink>; Département de microbiologie-infectiologiee et d'immunologie, Centres PROTEO et ARThrite, Faculté de Médecine, Université Laval, Quebec City, QC, G1V 0A6, Canada.; Axe Maladies infectieuses et immunitaires, Centre de recherche du CHU de Québec, Université Laval, Quebec City, QC, G1V 4G2, Canada.<br /><searchLink fieldCode="AU" term="%22Pelletier+J%22">Pelletier J</searchLink>; Axe Maladies infectieuses et immunitaires, Centre de recherche du CHU de Québec, Université Laval, Quebec City, QC, G1V 4G2, Canada.<br /><searchLink fieldCode="AU" term="%22Sévigny+J%22">Sévigny J</searchLink>; Département de microbiologie-infectiologiee et d'immunologie, Centres PROTEO et ARThrite, Faculté de Médecine, Université Laval, Quebec City, QC, G1V 0A6, Canada.; Axe Maladies infectieuses et immunitaires, Centre de recherche du CHU de Québec, Université Laval, Quebec City, QC, G1V 4G2, Canada.<br /><searchLink fieldCode="AU" term="%22Muhammad+M%22">Muhammad M</searchLink>; CAS Key Laboratory of Ion-Beam Bioengineering, Institute of Intelligent Machines, Hefei Institutes of Physical Science, Chinese Academy of Sciences, Hefei, China.<br /><searchLink fieldCode="AU" term="%22Huang+Q%22">Huang Q</searchLink>; CAS Key Laboratory of Ion-Beam Bioengineering, Institute of Intelligent Machines, Hefei Institutes of Physical Science, Chinese Academy of Sciences, Hefei, China.; Science Island Branch of Graduate School, University of Science and Technology of China, Hefei, China.<br /><searchLink fieldCode="AU" term="%22Iqbal+J%22">Iqbal J</searchLink>; Centre for Advanced Drug Research, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, 22060, Pakistan. drjamshed@cuiatd.edu.pk.; Department of Chemistry, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, 22060, Pakistan. drjamshed@cuiatd.edu.pk.
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              Text: 2026 Feb 21
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