Minimal chemical modification enables alpha/beta radiolabeling of sacituzumab govitecan for targeted therapy in high grade serous ovarian cancer.

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Title: Minimal chemical modification enables alpha/beta radiolabeling of sacituzumab govitecan for targeted therapy in high grade serous ovarian cancer.
Authors: Loor A; Molecular Pharmacology Program, Memorial Sloan Kettering Cancer Center, New York, NY, USA., Mack KN; Molecular Pharmacology Program, Memorial Sloan Kettering Cancer Center, New York, NY, USA.; Department of Pharmacology, Weill Cornell Graduate School of Medical Sciences, Weill Cornell Medicine, New York, NY, USA., Bauer D; Molecular Pharmacology Program, Memorial Sloan Kettering Cancer Center, New York, NY, USA., Ingham A; Molecular Pharmacology Program, Memorial Sloan Kettering Cancer Center, New York, NY, USA., Pratt EC; Molecular Pharmacology Program, Memorial Sloan Kettering Cancer Center, New York, NY, USA. edwin.pratt@stonybrookmedicine.edu.; Stony Brook University Cancer Center, Stony Brook, NY, USA. edwin.pratt@stonybrookmedicine.edu., Lewis JS; Molecular Pharmacology Program, Memorial Sloan Kettering Cancer Center, New York, NY, USA. lewisj2@mskcc.org.; Department of Pharmacology, Weill Cornell Graduate School of Medical Sciences, Weill Cornell Medicine, New York, NY, USA. lewisj2@mskcc.org.; Department of Radiology, Memorial Sloan Kettering Cancer Center, New York, NY, USA. lewisj2@mskcc.org.
Source: European journal of nuclear medicine and molecular imaging [Eur J Nucl Med Mol Imaging] 2026 Jun; Vol. 53 (7), pp. 4587-4596. Date of Electronic Publication: 2026 Feb 28.
Publication Type: Journal Article
Journal Info: Publisher: Springer-Verlag Berlin Country of Publication: Germany NLM ID: 101140988 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1619-7089 (Electronic) Linking ISSN: 16197070 NLM ISO Abbreviation: Eur J Nucl Med Mol Imaging Subsets: MEDLINE
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  Data: Minimal chemical modification enables alpha/beta radiolabeling of sacituzumab govitecan for targeted therapy in high grade serous ovarian cancer.
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  Data: <searchLink fieldCode="AU" term="%22Loor+A%22">Loor A</searchLink>; Molecular Pharmacology Program, Memorial Sloan Kettering Cancer Center, New York, NY, USA.<br /><searchLink fieldCode="AU" term="%22Mack+KN%22">Mack KN</searchLink>; Molecular Pharmacology Program, Memorial Sloan Kettering Cancer Center, New York, NY, USA.; Department of Pharmacology, Weill Cornell Graduate School of Medical Sciences, Weill Cornell Medicine, New York, NY, USA.<br /><searchLink fieldCode="AU" term="%22Bauer+D%22">Bauer D</searchLink>; Molecular Pharmacology Program, Memorial Sloan Kettering Cancer Center, New York, NY, USA.<br /><searchLink fieldCode="AU" term="%22Ingham+A%22">Ingham A</searchLink>; Molecular Pharmacology Program, Memorial Sloan Kettering Cancer Center, New York, NY, USA.<br /><searchLink fieldCode="AU" term="%22Pratt+EC%22">Pratt EC</searchLink>; Molecular Pharmacology Program, Memorial Sloan Kettering Cancer Center, New York, NY, USA. edwin.pratt@stonybrookmedicine.edu.; Stony Brook University Cancer Center, Stony Brook, NY, USA. edwin.pratt@stonybrookmedicine.edu.<br /><searchLink fieldCode="AU" term="%22Lewis+JS%22">Lewis JS</searchLink>; Molecular Pharmacology Program, Memorial Sloan Kettering Cancer Center, New York, NY, USA. lewisj2@mskcc.org.; Department of Pharmacology, Weill Cornell Graduate School of Medical Sciences, Weill Cornell Medicine, New York, NY, USA. lewisj2@mskcc.org.; Department of Radiology, Memorial Sloan Kettering Cancer Center, New York, NY, USA. lewisj2@mskcc.org.
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  Data: <searchLink fieldCode="JN" term="%22101140988%22">European journal of nuclear medicine and molecular imaging</searchLink> [Eur J Nucl Med Mol Imaging] 2026 Jun; Vol. 53 (7), pp. 4587-4596. <i>Date of Electronic Publication: </i>2026 Feb 28.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Springer-Verlag+Berlin%22">Springer-Verlag Berlin </searchLink><i>Country of Publication: </i>Germany <i>NLM ID: </i>101140988 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1619-7089 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2216197070%22">16197070 </searchLink><i>NLM ISO Abbreviation: </i>Eur J Nucl Med Mol Imaging <i>Subsets: </i>MEDLINE
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        Value: 10.1007/s00259-026-07820-7
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        Text: English
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        StartPage: 4587
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      – TitleFull: Minimal chemical modification enables alpha/beta radiolabeling of sacituzumab govitecan for targeted therapy in high grade serous ovarian cancer.
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              Text: 2026 Jun
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              Y: 2026
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