Novel indole-based sulfonate and sulfamate derivatives as potent and selective urease inhibitors targeting Helicobacter pylori: a promising therapeutic strategy.

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Title: Novel indole-based sulfonate and sulfamate derivatives as potent and selective urease inhibitors targeting Helicobacter pylori: a promising therapeutic strategy.
Authors: Khoder G; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates. gkhoder@sharjah.ac.ae.; Department of Pharmaceutics and Pharmaceutical Technology, College of Pharmacy, University of Sharjah, Sharjah, 27272, United Arab Emirates. gkhoder@sharjah.ac.ae., Mustafa EM; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates., Zaib S; Department of Basic and Applied Chemistry, Faculty of Science and Technology, University of Central Punjab, Lahore, 54590, Pakistan. sumera.zaib@ucp.edu.pk., Ravi A; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates., Shahin AI; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates., Zaraei SO; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates., Rana N; Department of Basic and Applied Chemistry, Faculty of Science and Technology, University of Central Punjab, Lahore, 54590, Pakistan., Anbar HS; Department of Pharmaceutical Sciences, College of Pharmacy, Dubai Medical University, Dubai, 19099, United Arab Emirates., Ali HS; Chemistry Research Laboratory, Department of Chemistry and the INEOS Oxford Institute for Antimicrobial Research, University of Oxford, 12 Mansfield Road, Oxford, OX1 3TA, UK., Qumar S; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates., Sebastian M; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates., Zein RA; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates., El-Gamal MI; Department of Medicinal Chemistry, College of Pharmacy, University of Sharjah, Sharjah, 27272, United Arab Emirates. drmelgamal2002@gmail.com.; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, 35516, Egypt. drmelgamal2002@gmail.com.
Source: Gut pathogens [Gut Pathog] 2026 Mar 04; Vol. 18 (1). Date of Electronic Publication: 2026 Mar 04.
Publication Type: Journal Article
Journal Info: Publisher: BioMed Central Country of Publication: England NLM ID: 101474263 Publication Model: Electronic Cited Medium: Print ISSN: 1757-4749 (Print) Linking ISSN: 17574749 NLM ISO Abbreviation: Gut Pathog Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
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  Data: Novel indole-based sulfonate and sulfamate derivatives as potent and selective urease inhibitors targeting Helicobacter pylori: a promising therapeutic strategy.
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  Data: <searchLink fieldCode="AU" term="%22Khoder+G%22">Khoder G</searchLink>; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates. gkhoder@sharjah.ac.ae.; Department of Pharmaceutics and Pharmaceutical Technology, College of Pharmacy, University of Sharjah, Sharjah, 27272, United Arab Emirates. gkhoder@sharjah.ac.ae.<br /><searchLink fieldCode="AU" term="%22Mustafa+EM%22">Mustafa EM</searchLink>; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates.<br /><searchLink fieldCode="AU" term="%22Zaib+S%22">Zaib S</searchLink>; Department of Basic and Applied Chemistry, Faculty of Science and Technology, University of Central Punjab, Lahore, 54590, Pakistan. sumera.zaib@ucp.edu.pk.<br /><searchLink fieldCode="AU" term="%22Ravi+A%22">Ravi A</searchLink>; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates.<br /><searchLink fieldCode="AU" term="%22Shahin+AI%22">Shahin AI</searchLink>; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates.<br /><searchLink fieldCode="AU" term="%22Zaraei+SO%22">Zaraei SO</searchLink>; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates.<br /><searchLink fieldCode="AU" term="%22Rana+N%22">Rana N</searchLink>; Department of Basic and Applied Chemistry, Faculty of Science and Technology, University of Central Punjab, Lahore, 54590, Pakistan.<br /><searchLink fieldCode="AU" term="%22Anbar+HS%22">Anbar HS</searchLink>; Department of Pharmaceutical Sciences, College of Pharmacy, Dubai Medical University, Dubai, 19099, United Arab Emirates.<br /><searchLink fieldCode="AU" term="%22Ali+HS%22">Ali HS</searchLink>; Chemistry Research Laboratory, Department of Chemistry and the INEOS Oxford Institute for Antimicrobial Research, University of Oxford, 12 Mansfield Road, Oxford, OX1 3TA, UK.<br /><searchLink fieldCode="AU" term="%22Qumar+S%22">Qumar S</searchLink>; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates.<br /><searchLink fieldCode="AU" term="%22Sebastian+M%22">Sebastian M</searchLink>; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates.<br /><searchLink fieldCode="AU" term="%22Zein+RA%22">Zein RA</searchLink>; Research Institute for Medical and Health Sciences, University of Sharjah, Sharjah, 27272, United Arab Emirates.<br /><searchLink fieldCode="AU" term="%22El-Gamal+MI%22">El-Gamal MI</searchLink>; Department of Medicinal Chemistry, College of Pharmacy, University of Sharjah, Sharjah, 27272, United Arab Emirates. drmelgamal2002@gmail.com.; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, 35516, Egypt. drmelgamal2002@gmail.com.
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  Data: <searchLink fieldCode="JN" term="%22101474263%22">Gut pathogens</searchLink> [Gut Pathog] 2026 Mar 04; Vol. 18 (1). <i>Date of Electronic Publication: </i>2026 Mar 04.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22BioMed+Central%22">BioMed Central </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>101474263 <i>Publication Model: </i>Electronic <i>Cited Medium: </i>Print <i>ISSN: </i>1757-4749 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2217574749%22">17574749 </searchLink><i>NLM ISO Abbreviation: </i>Gut Pathog <i>Subsets: </i>PubMed not MEDLINE
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              Text: 2026 Mar 04
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