Computational Design, Synthesis, and Evaluation of Stapled Peptide-Based Antagonists of the CGRP Receptor.
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| Title: | Computational Design, Synthesis, and Evaluation of Stapled Peptide-Based Antagonists of the CGRP Receptor. |
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| Authors: | Schofield AL; EaStChem School of Chemistry, The University of Edinburgh, Joseph Black Building, David Brewster Road, Edinburgh EH9 3FJ, U.K., Notari E; EaStChem School of Chemistry, The University of Edinburgh, Joseph Black Building, David Brewster Road, Edinburgh EH9 3FJ, U.K., Rožňovcová M; School of Pharmacy, University of Reading, Reading RG6 6AP, U.K., Cox KW; School of Pharmacy, University of Reading, Reading RG6 6AP, U.K., D'Aloisio V; School of Pharmacy and Biomolecular Sciences, Faculty of Science, Liverpool John Moores University, Liverpool L3 3AF, U.K., Steuer C; Institute of Pharmaceutical Sciences, ETH Zurich, HCI H401, Vladimir-Prelog-Weg 1-5/10, Zurich 8093, Switzerland., Michel J; EaStChem School of Chemistry, The University of Edinburgh, Joseph Black Building, David Brewster Road, Edinburgh EH9 3FJ, U.K., Cottrell GS; School of Pharmacy, University of Reading, Reading RG6 6AP, U.K., Coxon CR; EaStChem School of Chemistry, The University of Edinburgh, Joseph Black Building, David Brewster Road, Edinburgh EH9 3FJ, U.K. |
| Source: | Journal of medicinal chemistry [J Med Chem] 2026 Mar 26; Vol. 69 (6), pp. 7142-7159. Date of Electronic Publication: 2026 Mar 06. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 41789660 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Computational Design, Synthesis, and Evaluation of Stapled Peptide-Based Antagonists of the CGRP Receptor. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Schofield+AL%22">Schofield AL</searchLink>; EaStChem School of Chemistry, The University of Edinburgh, Joseph Black Building, David Brewster Road, Edinburgh EH9 3FJ, U.K.<br /><searchLink fieldCode="AU" term="%22Notari+E%22">Notari E</searchLink>; EaStChem School of Chemistry, The University of Edinburgh, Joseph Black Building, David Brewster Road, Edinburgh EH9 3FJ, U.K.<br /><searchLink fieldCode="AU" term="%22Rožňovcová+M%22">Rožňovcová M</searchLink>; School of Pharmacy, University of Reading, Reading RG6 6AP, U.K.<br /><searchLink fieldCode="AU" term="%22Cox+KW%22">Cox KW</searchLink>; School of Pharmacy, University of Reading, Reading RG6 6AP, U.K.<br /><searchLink fieldCode="AU" term="%22D'Aloisio+V%22">D'Aloisio V</searchLink>; School of Pharmacy and Biomolecular Sciences, Faculty of Science, Liverpool John Moores University, Liverpool L3 3AF, U.K.<br /><searchLink fieldCode="AU" term="%22Steuer+C%22">Steuer C</searchLink>; Institute of Pharmaceutical Sciences, ETH Zurich, HCI H401, Vladimir-Prelog-Weg 1-5/10, Zurich 8093, Switzerland.<br /><searchLink fieldCode="AU" term="%22Michel+J%22">Michel J</searchLink>; EaStChem School of Chemistry, The University of Edinburgh, Joseph Black Building, David Brewster Road, Edinburgh EH9 3FJ, U.K.<br /><searchLink fieldCode="AU" term="%22Cottrell+GS%22">Cottrell GS</searchLink>; School of Pharmacy, University of Reading, Reading RG6 6AP, U.K.<br /><searchLink fieldCode="AU" term="%22Coxon+CR%22">Coxon CR</searchLink>; EaStChem School of Chemistry, The University of Edinburgh, Joseph Black Building, David Brewster Road, Edinburgh EH9 3FJ, U.K. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 2026 Mar 26; Vol. 69 (6), pp. 7142-7159. <i>Date of Electronic Publication: </i>2026 Mar 06. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>9716531 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1520-4804 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200222623%22">00222623 </searchLink><i>NLM ISO Abbreviation: </i>J Med Chem <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=41789660 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/acs.jmedchem.5c03445 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 7142 Titles: – TitleFull: Computational Design, Synthesis, and Evaluation of Stapled Peptide-Based Antagonists of the CGRP Receptor. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Schofield AL – PersonEntity: Name: NameFull: Notari E – PersonEntity: Name: NameFull: Rožňovcová M – PersonEntity: Name: NameFull: Cox KW – PersonEntity: Name: NameFull: D'Aloisio V – PersonEntity: Name: NameFull: Steuer C – PersonEntity: Name: NameFull: Michel J – PersonEntity: Name: NameFull: Cottrell GS – PersonEntity: Name: NameFull: Coxon CR IsPartOfRelationships: – BibEntity: Dates: – D: 26 M: 03 Text: 2026 Mar 26 Type: published Y: 2026 Identifiers: – Type: issn-electronic Value: 1520-4804 Numbering: – Type: volume Value: 69 – Type: issue Value: 6 Titles: – TitleFull: Journal of medicinal chemistry Type: main |
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