N-aryl-N-acyl diamine derivatives as novel selective serotonin/norepinephrine transporter inhibitors for the treatment of premature ejaculation.

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Title: N-aryl-N-acyl diamine derivatives as novel selective serotonin/norepinephrine transporter inhibitors for the treatment of premature ejaculation.
Authors: Cui W; School of Pharmacy, Nantong University, 9 Seyuan Road, Nantong, 226019, China; Vigonvita Shanghai Co., Ltd., Shanghai, 201210, China., Nie K; Vigonvita Shanghai Co., Ltd., Shanghai, 201210, China., Jin F; Vigonvita Shanghai Co., Ltd., Shanghai, 201210, China., Li P; Vigonvita Shanghai Co., Ltd., Shanghai, 201210, China., Hou Q; Vigonvita Shanghai Co., Ltd., Shanghai, 201210, China., Hu T; Vigonvita Shanghai Co., Ltd., Shanghai, 201210, China., Tian G; Vigonvita Shanghai Co., Ltd., Shanghai, 201210, China., He Y; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China; University of Chinese Academy of Sciences, Beijing, 100049, China., Fan B; School of Pharmacy, Nantong University, 9 Seyuan Road, Nantong, 226019, China. Electronic address: fanboyi@ntu.edu.cn., Wang G; Vigonvita Shanghai Co., Ltd., Shanghai, 201210, China. Electronic address: guan.wang@vigonvita.cn., Shen J; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China; University of Chinese Academy of Sciences, Beijing, 100049, China.
Source: European journal of medicinal chemistry [Eur J Med Chem] 2026 Jun 05; Vol. 310, pp. 118771. Date of Electronic Publication: 2026 Mar 20.
Publication Type: Journal Article
Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1768-3254
DOI:10.1016/j.ejmech.2026.118771