Sequential Use of Trastuzumab Deruxtecan and Sacituzumab Govitecan in Patients with Breast Cancer: A Pharmacological Approach to Support the Clinical Rationale.

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Title: Sequential Use of Trastuzumab Deruxtecan and Sacituzumab Govitecan in Patients with Breast Cancer: A Pharmacological Approach to Support the Clinical Rationale.
Authors: Del Re M; Departmental Faculty of Medicine, Saint Camillus International University of Health and Medical Sciences, Rome, Italy.; Fondazione Policlinico Universitario IRCCS Agostino Gemelli, Rome, Italy., Inglese E; Unit of Clinical Chemistry, ASST Grande Ospedale Metropolitano, Niguarda, Milan, Italy., Bria E; Fondazione Policlinico Universitario IRCCS Agostino Gemelli, Rome, Italy.; Università Cattolica del Sacro Cuore, Rome, Italy., Blok EJ; Department of Medical Oncology, Leiden University Medical Center, Leiden, The Netherlands., Mathijssen RHJ; Department of Medical Oncology, Erasmus MC Cancer Institute, Erasmus University Medical Center, Rotterdam, The Netherlands., Curigliano G; Division of Development of New Drugs for Innovative Therapies, European Institute of Oncology IRCCS, Milan, Italy.; Department of Oncology and Hemato-Oncology, University of Milan 'La Statale', 7, Via Festa del Perdono, 20122, Milan, Italy., Danesi R; Department of Oncology and Hemato-Oncology, University of Milan 'La Statale', 7, Via Festa del Perdono, 20122, Milan, Italy. romano.danesi@unimi.it.
Source: Drugs [Drugs] 2026 Jun; Vol. 86 (6), pp. 871-885. Date of Electronic Publication: 2026 Apr 03.
Publication Type: Journal Article; Review
Journal Info: Publisher: Adis, Springer International Country of Publication: New Zealand NLM ID: 7600076 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1179-1950 (Electronic) Linking ISSN: 00126667 NLM ISO Abbreviation: Drugs Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Sequential Use of Trastuzumab Deruxtecan and Sacituzumab Govitecan in Patients with Breast Cancer: A Pharmacological Approach to Support the Clinical Rationale.
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  Data: <searchLink fieldCode="AU" term="%22Del+Re+M%22">Del Re M</searchLink>; Departmental Faculty of Medicine, Saint Camillus International University of Health and Medical Sciences, Rome, Italy.; Fondazione Policlinico Universitario IRCCS Agostino Gemelli, Rome, Italy.<br /><searchLink fieldCode="AU" term="%22Inglese+E%22">Inglese E</searchLink>; Unit of Clinical Chemistry, ASST Grande Ospedale Metropolitano, Niguarda, Milan, Italy.<br /><searchLink fieldCode="AU" term="%22Bria+E%22">Bria E</searchLink>; Fondazione Policlinico Universitario IRCCS Agostino Gemelli, Rome, Italy.; Università Cattolica del Sacro Cuore, Rome, Italy.<br /><searchLink fieldCode="AU" term="%22Blok+EJ%22">Blok EJ</searchLink>; Department of Medical Oncology, Leiden University Medical Center, Leiden, The Netherlands.<br /><searchLink fieldCode="AU" term="%22Mathijssen+RHJ%22">Mathijssen RHJ</searchLink>; Department of Medical Oncology, Erasmus MC Cancer Institute, Erasmus University Medical Center, Rotterdam, The Netherlands.<br /><searchLink fieldCode="AU" term="%22Curigliano+G%22">Curigliano G</searchLink>; Division of Development of New Drugs for Innovative Therapies, European Institute of Oncology IRCCS, Milan, Italy.; Department of Oncology and Hemato-Oncology, University of Milan 'La Statale', 7, Via Festa del Perdono, 20122, Milan, Italy.<br /><searchLink fieldCode="AU" term="%22Danesi+R%22">Danesi R</searchLink>; Department of Oncology and Hemato-Oncology, University of Milan 'La Statale', 7, Via Festa del Perdono, 20122, Milan, Italy. romano.danesi@unimi.it.
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      – TitleFull: Sequential Use of Trastuzumab Deruxtecan and Sacituzumab Govitecan in Patients with Breast Cancer: A Pharmacological Approach to Support the Clinical Rationale.
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              Text: 2026 Jun
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