A penicillin-binding protein inhibitor series to target drug-resistant Neisseria gonorrhoeae.

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Title: A penicillin-binding protein inhibitor series to target drug-resistant Neisseria gonorrhoeae.
Authors: Uehara T; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA. tsuyoshi.uehara@gmail.com., Zulli AL; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Miller B; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Avery LM; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Boyd SA; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Chatwin CL; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Chu GH; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Drager AS; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Edwards M; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Emeigh Hart SG; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Line NJ; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Myers CL; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Rongala G; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Stevenson A; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Uehara K; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Yi F; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Wang B; BioDuro-Sundia, Beijing, China., Liu Z; BioDuro-Sundia, Beijing, China., Wang M; BioDuro-Sundia, Beijing, China., Zhao Z; BioDuro-Sundia, Beijing, China., Zhou X; BioDuro-Sundia, Beijing, China., Zhao H; BioDuro-Sundia, Beijing, China., Stratton CM; Department of Biochemistry and Molecular Biology, University of South Alabama, Mobile, AL, USA., Bala S; Department of Biochemistry and Molecular Biology, University of South Alabama, Mobile, AL, USA., Davies C; Department of Biochemistry and Molecular Biology, University of South Alabama, Mobile, AL, USA., Tkavc R; Henry M. Jackson Foundation for the Advancement of Military Medicine, Bethesda, MD, USA.; Department of Microbiology and Immunology, Uniformed Services University of the Health Sciences, Bethesda, MD, USA., Jerse AE; Department of Microbiology and Immunology, Uniformed Services University of the Health Sciences, Bethesda, MD, USA., Pevear DC; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.; Spring Mill Pharma Inc., Malvern, PA, USA., Burns CJ; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Daigle DM; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA., Condon SM; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA. stephencondon3418@gmail.com.
Source: Nature microbiology [Nat Microbiol] 2026 May; Vol. 11 (5), pp. 1348-1360. Date of Electronic Publication: 2026 Apr 08.
Publication Type: Journal Article
Journal Info: Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101674869 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2058-5276 (Electronic) Linking ISSN: 20585276 NLM ISO Abbreviation: Nat Microbiol Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: A penicillin-binding protein inhibitor series to target drug-resistant Neisseria gonorrhoeae.
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  Data: <searchLink fieldCode="AU" term="%22Uehara+T%22">Uehara T</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA. tsuyoshi.uehara@gmail.com.<br /><searchLink fieldCode="AU" term="%22Zulli+AL%22">Zulli AL</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Miller+B%22">Miller B</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Avery+LM%22">Avery LM</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Boyd+SA%22">Boyd SA</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Chatwin+CL%22">Chatwin CL</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Chu+GH%22">Chu GH</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Drager+AS%22">Drager AS</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Edwards+M%22">Edwards M</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Emeigh+Hart+SG%22">Emeigh Hart SG</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Line+NJ%22">Line NJ</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Myers+CL%22">Myers CL</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Rongala+G%22">Rongala G</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Stevenson+A%22">Stevenson A</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Uehara+K%22">Uehara K</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Yi+F%22">Yi F</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Wang+B%22">Wang B</searchLink>; BioDuro-Sundia, Beijing, China.<br /><searchLink fieldCode="AU" term="%22Liu+Z%22">Liu Z</searchLink>; BioDuro-Sundia, Beijing, China.<br /><searchLink fieldCode="AU" term="%22Wang+M%22">Wang M</searchLink>; BioDuro-Sundia, Beijing, China.<br /><searchLink fieldCode="AU" term="%22Zhao+Z%22">Zhao Z</searchLink>; BioDuro-Sundia, Beijing, China.<br /><searchLink fieldCode="AU" term="%22Zhou+X%22">Zhou X</searchLink>; BioDuro-Sundia, Beijing, China.<br /><searchLink fieldCode="AU" term="%22Zhao+H%22">Zhao H</searchLink>; BioDuro-Sundia, Beijing, China.<br /><searchLink fieldCode="AU" term="%22Stratton+CM%22">Stratton CM</searchLink>; Department of Biochemistry and Molecular Biology, University of South Alabama, Mobile, AL, USA.<br /><searchLink fieldCode="AU" term="%22Bala+S%22">Bala S</searchLink>; Department of Biochemistry and Molecular Biology, University of South Alabama, Mobile, AL, USA.<br /><searchLink fieldCode="AU" term="%22Davies+C%22">Davies C</searchLink>; Department of Biochemistry and Molecular Biology, University of South Alabama, Mobile, AL, USA.<br /><searchLink fieldCode="AU" term="%22Tkavc+R%22">Tkavc R</searchLink>; Henry M. Jackson Foundation for the Advancement of Military Medicine, Bethesda, MD, USA.; Department of Microbiology and Immunology, Uniformed Services University of the Health Sciences, Bethesda, MD, USA.<br /><searchLink fieldCode="AU" term="%22Jerse+AE%22">Jerse AE</searchLink>; Department of Microbiology and Immunology, Uniformed Services University of the Health Sciences, Bethesda, MD, USA.<br /><searchLink fieldCode="AU" term="%22Pevear+DC%22">Pevear DC</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.; Spring Mill Pharma Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Burns+CJ%22">Burns CJ</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Daigle+DM%22">Daigle DM</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA.<br /><searchLink fieldCode="AU" term="%22Condon+SM%22">Condon SM</searchLink>; Venatorx Pharmaceuticals, Inc., Malvern, PA, USA. stephencondon3418@gmail.com.
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  Data: <searchLink fieldCode="JN" term="%22101674869%22">Nature microbiology</searchLink> [Nat Microbiol] 2026 May; Vol. 11 (5), pp. 1348-1360. <i>Date of Electronic Publication: </i>2026 Apr 08.
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