Discovery and characterization of a covalent inhibitor of New Delhi metallo β-lactamase.
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| Title: | Discovery and characterization of a covalent inhibitor of New Delhi metallo β-lactamase. |
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| Authors: | Rivera DD; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States., Schroeder JM; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States., Walker JN; Department of Chemistry, The University of Texas at Austin, Austin, TX, 78712, United States., Bashyal A; Department of Chemistry, The University of Texas at Austin, Austin, TX, 78712, United States., Iyer AG; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States., Lee RH; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States., Melkonian TR; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States., Brodbelt JS; Department of Chemistry, The University of Texas at Austin, Austin, TX, 78712, United States., Fast W; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States., Whitman CP; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States. Electronic address: whitman@austin.utexas.edu. |
| Source: | Archives of biochemistry and biophysics [Arch Biochem Biophys] 2026 Jul; Vol. 781, pp. 110805. Date of Electronic Publication: 2026 Apr 07. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Elsevier Country of Publication: United States NLM ID: 0372430 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1096-0384 (Electronic) Linking ISSN: 00039861 NLM ISO Abbreviation: Arch Biochem Biophys Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 41956364 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Discovery and characterization of a covalent inhibitor of New Delhi metallo β-lactamase. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Rivera+DD%22">Rivera DD</searchLink>; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Schroeder+JM%22">Schroeder JM</searchLink>; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Walker+JN%22">Walker JN</searchLink>; Department of Chemistry, The University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Bashyal+A%22">Bashyal A</searchLink>; Department of Chemistry, The University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Iyer+AG%22">Iyer AG</searchLink>; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Lee+RH%22">Lee RH</searchLink>; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Melkonian+TR%22">Melkonian TR</searchLink>; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Brodbelt+JS%22">Brodbelt JS</searchLink>; Department of Chemistry, The University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Fast+W%22">Fast W</searchLink>; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Whitman+CP%22">Whitman CP</searchLink>; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States. Electronic address: whitman@austin.utexas.edu. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%220372430%22">Archives of biochemistry and biophysics</searchLink> [Arch Biochem Biophys] 2026 Jul; Vol. 781, pp. 110805. <i>Date of Electronic Publication: </i>2026 Apr 07. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier%22">Elsevier </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>0372430 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1096-0384 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200039861%22">00039861 </searchLink><i>NLM ISO Abbreviation: </i>Arch Biochem Biophys <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=41956364 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.abb.2026.110805 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 110805 Titles: – TitleFull: Discovery and characterization of a covalent inhibitor of New Delhi metallo β-lactamase. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Rivera DD – PersonEntity: Name: NameFull: Schroeder JM – PersonEntity: Name: NameFull: Walker JN – PersonEntity: Name: NameFull: Bashyal A – PersonEntity: Name: NameFull: Iyer AG – PersonEntity: Name: NameFull: Lee RH – PersonEntity: Name: NameFull: Melkonian TR – PersonEntity: Name: NameFull: Brodbelt JS – PersonEntity: Name: NameFull: Fast W – PersonEntity: Name: NameFull: Whitman CP IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 07 Text: 2026 Jul Type: published Y: 2026 Identifiers: – Type: issn-electronic Value: 1096-0384 Numbering: – Type: volume Value: 781 Titles: – TitleFull: Archives of biochemistry and biophysics Type: main |
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