Discovery and characterization of a covalent inhibitor of New Delhi metallo β-lactamase.

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Title: Discovery and characterization of a covalent inhibitor of New Delhi metallo β-lactamase.
Authors: Rivera DD; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States., Schroeder JM; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States., Walker JN; Department of Chemistry, The University of Texas at Austin, Austin, TX, 78712, United States., Bashyal A; Department of Chemistry, The University of Texas at Austin, Austin, TX, 78712, United States., Iyer AG; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States., Lee RH; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States., Melkonian TR; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States., Brodbelt JS; Department of Chemistry, The University of Texas at Austin, Austin, TX, 78712, United States., Fast W; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States., Whitman CP; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States. Electronic address: whitman@austin.utexas.edu.
Source: Archives of biochemistry and biophysics [Arch Biochem Biophys] 2026 Jul; Vol. 781, pp. 110805. Date of Electronic Publication: 2026 Apr 07.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Country of Publication: United States NLM ID: 0372430 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1096-0384 (Electronic) Linking ISSN: 00039861 NLM ISO Abbreviation: Arch Biochem Biophys Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Discovery and characterization of a covalent inhibitor of New Delhi metallo β-lactamase.
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  Data: <searchLink fieldCode="AU" term="%22Rivera+DD%22">Rivera DD</searchLink>; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Schroeder+JM%22">Schroeder JM</searchLink>; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Walker+JN%22">Walker JN</searchLink>; Department of Chemistry, The University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Bashyal+A%22">Bashyal A</searchLink>; Department of Chemistry, The University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Iyer+AG%22">Iyer AG</searchLink>; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Lee+RH%22">Lee RH</searchLink>; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Melkonian+TR%22">Melkonian TR</searchLink>; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Brodbelt+JS%22">Brodbelt JS</searchLink>; Department of Chemistry, The University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Fast+W%22">Fast W</searchLink>; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States.<br /><searchLink fieldCode="AU" term="%22Whitman+CP%22">Whitman CP</searchLink>; Division of Chemical Biology and Medicinal Chemistry, College of Pharmacy, University of Texas at Austin, Austin, TX, 78712, United States. Electronic address: whitman@austin.utexas.edu.
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              Text: 2026 Jul
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