Towards the targeted protein degradation of CK2: design and synthesis of CAM4066-based PROTACs.
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| Title: | Towards the targeted protein degradation of CK2: design and synthesis of CAM4066-based PROTACs. |
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| Authors: | Day-Riley S; Yusuf Hamied Department of Chemistry, University of Cambridge, Lensfield Road, CB2 1EW, Cambridge, United Kingdom., Krajcovicova S; Yusuf Hamied Department of Chemistry, University of Cambridge, Lensfield Road, CB2 1EW, Cambridge, United Kingdom.; Department of Organic Chemistry, Faculty of Science, Palacky University, Tr. 17. Listopadu 12, Olomouc, 77900, Czech Republic., Sokhal AR; Yusuf Hamied Department of Chemistry, University of Cambridge, Lensfield Road, CB2 1EW, Cambridge, United Kingdom., Venne JL; Yusuf Hamied Department of Chemistry, University of Cambridge, Lensfield Road, CB2 1EW, Cambridge, United Kingdom., Brear P; Department of Biochemistry, University of Cambridge, Tennis Court Road, Cambridge, CB2 1GA, United Kingdom., Hyvönen M; Department of Biochemistry, University of Cambridge, Tennis Court Road, Cambridge, CB2 1GA, United Kingdom., Whitehurst BC; Hit Discovery, Discovery Sciences, R&D, AstraZeneca, Cambridge, CB2 0AA, United Kingdom., Carroll JS; Cancer Research UK Cambridge Institute, Robinson Way, Cambridge, CB2 0RE, United Kingdom., Spring DR; Yusuf Hamied Department of Chemistry, University of Cambridge, Lensfield Road, CB2 1EW, Cambridge, United Kingdom. |
| Source: | Beilstein journal of organic chemistry [Beilstein J Org Chem] 2026 Apr 22; Vol. 22, pp. 611-619. Date of Electronic Publication: 2026 Apr 22 (Print Publication: 2026). |
| Publication Type: | Letter |
| Journal Info: | Publisher: Beilstein-Institut Country of Publication: Germany NLM ID: 101250746 Publication Model: eCollection Cited Medium: Print ISSN: 1860-5397 (Print) Linking ISSN: 18605397 NLM ISO Abbreviation: Beilstein J Org Chem Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
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