Hierarchical small molecule inhibition of MYST acetyltransferases.

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Title: Hierarchical small molecule inhibition of MYST acetyltransferases.
Authors: Chen X; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA., Castroverde A; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA., Perez M; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA., Holewinski R; Protein Characterization Laboratory, Frederick National Laboratory for Cancer Research, Leidos Biomedical Research, Frederick, Maryland, USA., Suazo KF; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA.; Protein Characterization Laboratory, Frederick National Laboratory for Cancer Research, Leidos Biomedical Research, Frederick, Maryland, USA., Karki R; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri, USA., Andresson T; Protein Characterization Laboratory, Frederick National Laboratory for Cancer Research, Leidos Biomedical Research, Frederick, Maryland, USA., Garcia BA; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri, USA., Meier JL; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA. jordan.meier@nih.gov.
Source: Nature communications [Nat Commun] 2026 May 13; Vol. 17 (1). Date of Electronic Publication: 2026 May 13.
Publication Type: Journal Article
Journal Info: Publisher: Nature Pub. Group Country of Publication: England NLM ID: 101528555 Publication Model: Electronic Cited Medium: Internet ISSN: 2041-1723 (Electronic) Linking ISSN: 20411723 NLM ISO Abbreviation: Nat Commun Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Hierarchical small molecule inhibition of MYST acetyltransferases.
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  Data: <searchLink fieldCode="AU" term="%22Chen+X%22">Chen X</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA.<br /><searchLink fieldCode="AU" term="%22Castroverde+A%22">Castroverde A</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA.<br /><searchLink fieldCode="AU" term="%22Perez+M%22">Perez M</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA.<br /><searchLink fieldCode="AU" term="%22Holewinski+R%22">Holewinski R</searchLink>; Protein Characterization Laboratory, Frederick National Laboratory for Cancer Research, Leidos Biomedical Research, Frederick, Maryland, USA.<br /><searchLink fieldCode="AU" term="%22Suazo+KF%22">Suazo KF</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA.; Protein Characterization Laboratory, Frederick National Laboratory for Cancer Research, Leidos Biomedical Research, Frederick, Maryland, USA.<br /><searchLink fieldCode="AU" term="%22Karki+R%22">Karki R</searchLink>; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri, USA.<br /><searchLink fieldCode="AU" term="%22Andresson+T%22">Andresson T</searchLink>; Protein Characterization Laboratory, Frederick National Laboratory for Cancer Research, Leidos Biomedical Research, Frederick, Maryland, USA.<br /><searchLink fieldCode="AU" term="%22Garcia+BA%22">Garcia BA</searchLink>; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri, USA.<br /><searchLink fieldCode="AU" term="%22Meier+JL%22">Meier JL</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA. jordan.meier@nih.gov.
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  Data: <searchLink fieldCode="JN" term="%22101528555%22">Nature communications</searchLink> [Nat Commun] 2026 May 13; Vol. 17 (1). <i>Date of Electronic Publication: </i>2026 May 13.
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        Value: 10.1038/s41467-026-70574-1
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              Text: 2026 May 13
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