Hierarchical small molecule inhibition of MYST acetyltransferases.
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| Title: | Hierarchical small molecule inhibition of MYST acetyltransferases. |
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| Authors: | Chen X; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA., Castroverde A; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA., Perez M; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA., Holewinski R; Protein Characterization Laboratory, Frederick National Laboratory for Cancer Research, Leidos Biomedical Research, Frederick, Maryland, USA., Suazo KF; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA.; Protein Characterization Laboratory, Frederick National Laboratory for Cancer Research, Leidos Biomedical Research, Frederick, Maryland, USA., Karki R; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri, USA., Andresson T; Protein Characterization Laboratory, Frederick National Laboratory for Cancer Research, Leidos Biomedical Research, Frederick, Maryland, USA., Garcia BA; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri, USA., Meier JL; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA. jordan.meier@nih.gov. |
| Source: | Nature communications [Nat Commun] 2026 May 13; Vol. 17 (1). Date of Electronic Publication: 2026 May 13. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Nature Pub. Group Country of Publication: England NLM ID: 101528555 Publication Model: Electronic Cited Medium: Internet ISSN: 2041-1723 (Electronic) Linking ISSN: 20411723 NLM ISO Abbreviation: Nat Commun Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 42129151 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Hierarchical small molecule inhibition of MYST acetyltransferases. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Chen+X%22">Chen X</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA.<br /><searchLink fieldCode="AU" term="%22Castroverde+A%22">Castroverde A</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA.<br /><searchLink fieldCode="AU" term="%22Perez+M%22">Perez M</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA.<br /><searchLink fieldCode="AU" term="%22Holewinski+R%22">Holewinski R</searchLink>; Protein Characterization Laboratory, Frederick National Laboratory for Cancer Research, Leidos Biomedical Research, Frederick, Maryland, USA.<br /><searchLink fieldCode="AU" term="%22Suazo+KF%22">Suazo KF</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA.; Protein Characterization Laboratory, Frederick National Laboratory for Cancer Research, Leidos Biomedical Research, Frederick, Maryland, USA.<br /><searchLink fieldCode="AU" term="%22Karki+R%22">Karki R</searchLink>; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri, USA.<br /><searchLink fieldCode="AU" term="%22Andresson+T%22">Andresson T</searchLink>; Protein Characterization Laboratory, Frederick National Laboratory for Cancer Research, Leidos Biomedical Research, Frederick, Maryland, USA.<br /><searchLink fieldCode="AU" term="%22Garcia+BA%22">Garcia BA</searchLink>; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, Missouri, USA.<br /><searchLink fieldCode="AU" term="%22Meier+JL%22">Meier JL</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland, USA. jordan.meier@nih.gov. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101528555%22">Nature communications</searchLink> [Nat Commun] 2026 May 13; Vol. 17 (1). <i>Date of Electronic Publication: </i>2026 May 13. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Nature+Pub%2E+Group%22">Nature Pub. Group </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>101528555 <i>Publication Model: </i>Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>2041-1723 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2220411723%22">20411723 </searchLink><i>NLM ISO Abbreviation: </i>Nat Commun <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=42129151 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1038/s41467-026-70574-1 Languages: – Code: eng Text: English Titles: – TitleFull: Hierarchical small molecule inhibition of MYST acetyltransferases. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Chen X – PersonEntity: Name: NameFull: Castroverde A – PersonEntity: Name: NameFull: Perez M – PersonEntity: Name: NameFull: Holewinski R – PersonEntity: Name: NameFull: Suazo KF – PersonEntity: Name: NameFull: Karki R – PersonEntity: Name: NameFull: Andresson T – PersonEntity: Name: NameFull: Garcia BA – PersonEntity: Name: NameFull: Meier JL IsPartOfRelationships: – BibEntity: Dates: – D: 13 M: 05 Text: 2026 May 13 Type: published Y: 2026 Identifiers: – Type: issn-electronic Value: 2041-1723 Numbering: – Type: volume Value: 17 – Type: issue Value: 1 Titles: – TitleFull: Nature communications Type: main |
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