CYP3A-Mediated Metabolism of Zastaprazan in Humans and Associated Drug-Drug Interactions.

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Title: CYP3A-Mediated Metabolism of Zastaprazan in Humans and Associated Drug-Drug Interactions.
Authors: Cao KJ; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.; University of Chinese Academy of Sciences, Beijing 100049, China., Fu L; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China., Sun YC; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China., Meng J; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China., Huang Q; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China., Deng DC; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China., Hu HT; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China., Han ZH; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China., Guo G; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China., Zhou X; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China.; School of Pharmacy, Fudan University, Shanghai 200433, China., Chen XY; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.; University of Chinese Academy of Sciences, Beijing 100049, China.
Source: Pharmaceutics [Pharmaceutics] 2026 Jun 10; Vol. 18 (6). Date of Electronic Publication: 2026 Jun 10.
Publication Type: Journal Article
Journal Info: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101534003 Publication Model: Electronic Cited Medium: Print ISSN: 1999-4923 (Print) Linking ISSN: 19994923 NLM ISO Abbreviation: Pharmaceutics Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
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  Data: CYP3A-Mediated Metabolism of Zastaprazan in Humans and Associated Drug-Drug Interactions.
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  Data: <searchLink fieldCode="AU" term="%22Cao+KJ%22">Cao KJ</searchLink>; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.; University of Chinese Academy of Sciences, Beijing 100049, China.<br /><searchLink fieldCode="AU" term="%22Fu+L%22">Fu L</searchLink>; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China.<br /><searchLink fieldCode="AU" term="%22Sun+YC%22">Sun YC</searchLink>; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.<br /><searchLink fieldCode="AU" term="%22Meng+J%22">Meng J</searchLink>; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.<br /><searchLink fieldCode="AU" term="%22Huang+Q%22">Huang Q</searchLink>; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China.<br /><searchLink fieldCode="AU" term="%22Deng+DC%22">Deng DC</searchLink>; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China.<br /><searchLink fieldCode="AU" term="%22Hu+HT%22">Hu HT</searchLink>; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China.<br /><searchLink fieldCode="AU" term="%22Han+ZH%22">Han ZH</searchLink>; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China.<br /><searchLink fieldCode="AU" term="%22Guo+G%22">Guo G</searchLink>; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.<br /><searchLink fieldCode="AU" term="%22Zhou+X%22">Zhou X</searchLink>; Livzon Pharmaceutical Group Inc., Zhuhai 519000, China.; School of Pharmacy, Fudan University, Shanghai 200433, China.<br /><searchLink fieldCode="AU" term="%22Chen+XY%22">Chen XY</searchLink>; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.; University of Chinese Academy of Sciences, Beijing 100049, China.
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  Data: <searchLink fieldCode="JN" term="%22101534003%22">Pharmaceutics</searchLink> [Pharmaceutics] 2026 Jun 10; Vol. 18 (6). <i>Date of Electronic Publication: </i>2026 Jun 10.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22MDPI%22">MDPI </searchLink><i>Country of Publication: </i>Switzerland <i>NLM ID: </i>101534003 <i>Publication Model: </i>Electronic <i>Cited Medium: </i>Print <i>ISSN: </i>1999-4923 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2219994923%22">19994923 </searchLink><i>NLM ISO Abbreviation: </i>Pharmaceutics <i>Subsets: </i>PubMed not MEDLINE
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        Value: 10.3390/pharmaceutics18060718
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        Text: English
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      – TitleFull: CYP3A-Mediated Metabolism of Zastaprazan in Humans and Associated Drug-Drug Interactions.
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            – D: 10
              M: 06
              Text: 2026 Jun 10
              Type: published
              Y: 2026
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