Next-generation chemogenetic inhibition using a brain-permeant non-prescription agent.

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Title: Next-generation chemogenetic inhibition using a brain-permeant non-prescription agent.
Authors: Devenish SO; UCL Queen Square Institute of Neurology, University College London, London, UK. s.o.devenish@gmail.com., Patel SD; UCL Queen Square Institute of Neurology, University College London, London, UK., Ussingkær LV; UCL Queen Square Institute of Neurology, University College London, London, UK., Almeida Silva LF; UCL Queen Square Institute of Neurology, University College London, London, UK., Goff O; UCL Queen Square Institute of Neurology, University College London, London, UK., Richardson A; UCL Queen Square Institute of Neurology, University College London, London, UK., Mobbs JI; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia., Venugopal H; Ramaciotti Centre for Cryo-Electron Microscopy, Monash University, Clayton, Australia., Thal DM; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia. David.Thal@monash.edu.; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia. David.Thal@monash.edu., Kullmann DM; UCL Queen Square Institute of Neurology, University College London, London, UK. d.kullmann@ucl.ac.uk.
Source: Signal transduction and targeted therapy [Signal Transduct Target Ther] 2026 Jul 03; Vol. 11 (1). Date of Electronic Publication: 2026 Jul 03.
Publication Type: Journal Article
Journal Info: Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101676423 Publication Model: Electronic Cited Medium: Internet ISSN: 2059-3635 (Electronic) Linking ISSN: 20593635 NLM ISO Abbreviation: Signal Transduct Target Ther Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:2059-3635
DOI:10.1038/s41392-026-02865-4