Alpha-Particle Therapy with an Actinium-225 Labeled Bivalent Inhibitor of Prostate-Specific Membrane Antigen is Therapeutically Efficacious in a Mouse Model of Prostate Cancer.

Saved in:
Bibliographic Details
Title: Alpha-Particle Therapy with an Actinium-225 Labeled Bivalent Inhibitor of Prostate-Specific Membrane Antigen is Therapeutically Efficacious in a Mouse Model of Prostate Cancer.
Authors: Morgan KA; School of Chemistry and Bio21 Molecular Science and Biotechnology Institute, University of Melbourne, Melbourne, 3010 Victoria, Australia., Grieve ML; Australian Institute for Bioengineering and Nanotechnology, the University of Queensland, Brisbane, QLD 4072, Australia.; ARC Research Hub for Advanced Manufacture of Targeted Radiopharmaceuticals (AMTAR), the University of Queensland, Brisbane, QLD 4072, Australia., Akhter DT; Australian Institute for Bioengineering and Nanotechnology, the University of Queensland, Brisbane, QLD 4072, Australia.; ARC Research Hub for Advanced Manufacture of Targeted Radiopharmaceuticals (AMTAR), the University of Queensland, Brisbane, QLD 4072, Australia., Lange JL; Clarity Pharmaceuticals Ltd., National Innovation Centre, 4 Cornwallis Street, Eveleigh, New South Wales 2042, Australia., Harris MJ; Clarity Pharmaceuticals Ltd., National Innovation Centre, 4 Cornwallis Street, Eveleigh, New South Wales 2042, Australia., Thurecht KJ; Australian Institute for Bioengineering and Nanotechnology, the University of Queensland, Brisbane, QLD 4072, Australia.; ARC Research Hub for Advanced Manufacture of Targeted Radiopharmaceuticals (AMTAR), the University of Queensland, Brisbane, QLD 4072, Australia., Paterson BM; Australian Institute for Bioengineering and Nanotechnology, the University of Queensland, Brisbane, QLD 4072, Australia.; ARC Research Hub for Advanced Manufacture of Targeted Radiopharmaceuticals (AMTAR), the University of Queensland, Brisbane, QLD 4072, Australia., Donnelly PS; School of Chemistry and Bio21 Molecular Science and Biotechnology Institute, University of Melbourne, Melbourne, 3010 Victoria, Australia.
Source: Journal of medicinal chemistry [J Med Chem] 2026 Jul 23; Vol. 69 (14), pp. 17462-17472. Date of Electronic Publication: 2026 Jul 04.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1520-4804
DOI:10.1021/acs.jmedchem.6c01378