From dual norepinephrine-dopamine reuptake inhibition to selective dopamine reuptake inhibitors: a case of aromatically substituted N,2-cyclopentylamines.
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| Title: | From dual norepinephrine-dopamine reuptake inhibition to selective dopamine reuptake inhibitors: a case of aromatically substituted N,2-cyclopentylamines. |
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| Authors: | Dilweg MA; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl., Jespers W; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl.; Department of Medicinal Chemistry, Photopharmacology and Imaging, Groningen Research Institute of Pharmacy (GRIP), Faculty of Science and Engineering Antonius Deusinglaan 1 9713 AV Groningen The Netherlands., Kasture AS; Institute of Pharmacology, Medical University of Vienna Vienna Austria.; Department of Neurosciences and Developmental Biology, University of Vienna Vienna Austria., Liu R; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl., Mocking TAM; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl., van der Ploeg JG; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl., Baselier AMM; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl., van Westen GJP; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl., Hummel T; Department of Neurosciences and Developmental Biology, University of Vienna Vienna Austria., Sucic S; Institute of Pharmacology, Medical University of Vienna Vienna Austria., IJzerman AP; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl., Heitman LH; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl.; Oncode Institute Leiden The Netherlands., van der Es D; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl. |
| Source: | RSC medicinal chemistry [RSC Med Chem] 2026 Jun 24; Vol. 17 (7), pp. 3447-3462. Date of Electronic Publication: 2026 Jun 24 (Print Publication: 2026). |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 101759460 Publication Model: eCollection Cited Medium: Internet ISSN: 2632-8682 (Electronic) Linking ISSN: 26328682 NLM ISO Abbreviation: RSC Med Chem Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
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