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Synthesis and biological evaluation of the 1,5-diarylpyrazole class of cyclooxygenase-2 inhibitors: identification of 4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]benze nesulfonamide (SC-58635, celecoxib).

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Title: Synthesis and biological evaluation of the 1,5-diarylpyrazole class of cyclooxygenase-2 inhibitors: identification of 4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]benze nesulfonamide (SC-58635, celecoxib).
Authors: Penning TD; Department of Chemistry, Searle Research and Development, Skokie, Illinois 60077, USA., Talley JJ, Bertenshaw SR, Carter JS, Collins PW, Docter S, Graneto MJ, Lee LF, Malecha JW, Miyashiro JM, Rogers RS, Rogier DJ, Yu SS, AndersonGD, Burton EG, Cogburn JN, Gregory SA, Koboldt CM, Perkins WE, Seibert K, Veenhuizen AW, Zhang YY, Isakson PC
Source: Journal of medicinal chemistry [J Med Chem] 1997 Apr 25; Vol. 40 (9), pp. 1347-65.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print Cited Medium: Print ISSN: 0022-2623 (Print) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Synthesis and biological evaluation of the 1,5-diarylpyrazole class of cyclooxygenase-2 inhibitors: identification of 4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]benze nesulfonamide (SC-58635, celecoxib).
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  Data: <searchLink fieldCode="AU" term="%22Penning+TD%22">Penning TD</searchLink>; Department of Chemistry, Searle Research and Development, Skokie, Illinois 60077, USA.<br /><searchLink fieldCode="AU" term="%22Talley+JJ%22">Talley JJ</searchLink><br /><searchLink fieldCode="AU" term="%22Bertenshaw+SR%22">Bertenshaw SR</searchLink><br /><searchLink fieldCode="AU" term="%22Carter+JS%22">Carter JS</searchLink><br /><searchLink fieldCode="AU" term="%22Collins+PW%22">Collins PW</searchLink><br /><searchLink fieldCode="AU" term="%22Docter+S%22">Docter S</searchLink><br /><searchLink fieldCode="AU" term="%22Graneto+MJ%22">Graneto MJ</searchLink><br /><searchLink fieldCode="AU" term="%22Lee+LF%22">Lee LF</searchLink><br /><searchLink fieldCode="AU" term="%22Malecha+JW%22">Malecha JW</searchLink><br /><searchLink fieldCode="AU" term="%22Miyashiro+JM%22">Miyashiro JM</searchLink><br /><searchLink fieldCode="AU" term="%22Rogers+RS%22">Rogers RS</searchLink><br /><searchLink fieldCode="AU" term="%22Rogier+DJ%22">Rogier DJ</searchLink><br /><searchLink fieldCode="AU" term="%22Yu+SS%22">Yu SS</searchLink><br /><searchLink fieldCode="AU" term="%22AndersonGD%22">AndersonGD</searchLink><br /><searchLink fieldCode="AU" term="%22Burton+EG%22">Burton EG</searchLink><br /><searchLink fieldCode="AU" term="%22Cogburn+JN%22">Cogburn JN</searchLink><br /><searchLink fieldCode="AU" term="%22Gregory+SA%22">Gregory SA</searchLink><br /><searchLink fieldCode="AU" term="%22Koboldt+CM%22">Koboldt CM</searchLink><br /><searchLink fieldCode="AU" term="%22Perkins+WE%22">Perkins WE</searchLink><br /><searchLink fieldCode="AU" term="%22Seibert+K%22">Seibert K</searchLink><br /><searchLink fieldCode="AU" term="%22Veenhuizen+AW%22">Veenhuizen AW</searchLink><br /><searchLink fieldCode="AU" term="%22Zhang+YY%22">Zhang YY</searchLink><br /><searchLink fieldCode="AU" term="%22Isakson+PC%22">Isakson PC</searchLink>
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  Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 1997 Apr 25; Vol. 40 (9), pp. 1347-65.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>9716531 <i>Publication Model: </i>Print <i>Cited Medium: </i>Print <i>ISSN: </i>0022-2623 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200222623%22">00222623 </searchLink><i>NLM ISO Abbreviation: </i>J Med Chem <i>Subsets: </i>MEDLINE
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