Novel Analogues of (R)-5-(Methylamino)-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (Sumanirole) Provide Clues to Dopamine D2/D3 Receptor Agonist Selectivity.

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Title: Novel Analogues of (R)-5-(Methylamino)-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (Sumanirole) Provide Clues to Dopamine D2/D3 Receptor Agonist Selectivity.
Authors: Mu-Fa Zou1, Keck, Thomas M.1, Kumar, Vivek1, Donthamsetti, Prashant2, Michino, Mayako3, Burzynski, Caitlin1, Schweppe, Catherine1, Bonifazi, Alessandro1, Free, R. Benjamin4, Sibley, David R.4, Janowsky, Aaron5,6, Lei Shi7, Javitch, Jonathan A.2,8, Newman, Amy Hauck1 anewman@intra.nida.nih.gov
Source: Journal of Medicinal Chemistry. 4/14/2016, Vol. 59 Issue 7, p2973-2988. 16p.
Database: Academic Search Ultimate
Description
ISSN:00222623
DOI:10.1021/acs.jmedchem.5b01612