Structure-based design and synthesis of 2,4-diaminopyrimidines as EGFR L858R/T790M selective inhibitors for NSCLC.

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Bibliographic Details
Title: Structure-based design and synthesis of 2,4-diaminopyrimidines as EGFR L858R/T790M selective inhibitors for NSCLC.
Authors: Chen, Lingfeng1,2, Fu, Weitao2, Feng, Chen2, Qu, Rong3, Tong, Linjiang3, Zheng, Lulu2, Fang, Bo2, Qiu, Yinda2, Hu, Jie2, Cai, Yuepiao2, Feng, Jianpeng2, Xie, Hua3, Ding, Jian3 jding@simm.ac.cn, Liu, Zhiguo2 lzgcnu@163.com, Liang, Guang1,2 wzmcliangguang@163.com
Source: European Journal of Medicinal Chemistry. Nov2017, Vol. 140, p510-527. 18p.
Database: Academic Search Ultimate
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