Discovery of Trifluoromethyl Glycol Carbamates as Potent and Selective Covalent Monoacylglycerol Lipase (MAGL) Inhibitors for Treatment of Neuroinflammation.
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| Title: | Discovery of Trifluoromethyl Glycol Carbamates as Potent and Selective Covalent Monoacylglycerol Lipase (MAGL) Inhibitors for Treatment of Neuroinflammation. |
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| Authors: | McAllister, Laura A.1 laura.mcallister@pfizer.com, Butler, Christopher R.1, Mente, Scot1, O'Neil, Steven V.2, Fonseca, Kari R.1, Piro, Justin R.1, Cianfrogna, Julie A.2, Foley, Timothy L.2, Gilbert, Adam M.2, Harris, Anthony R.2, Helal, Christopher J.2, Johnson, Douglas S.1, Montgomery, Justin I.2, Nason, Deane M.2, Noell, Stephen2, Pandit, Jayvardhan2, Rogers, Bruce N.1, Samad, Tarek A.1, Shaffer, Christopher L.1, Silva, Rafael G. da2 |
| Source: | Journal of Medicinal Chemistry. 4/12/2018, Vol. 61 Issue 7, p3008-3026. 19p. |
| Database: | Academic Search Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: asn DbLabel: Academic Search Ultimate An: 129283375 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=129283375 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/acs.jmedchem.8b00070 Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 19 StartPage: 3008 Titles: – TitleFull: Discovery of Trifluoromethyl Glycol Carbamates as Potent and Selective Covalent Monoacylglycerol Lipase (MAGL) Inhibitors for Treatment of Neuroinflammation. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: McAllister, Laura A. – PersonEntity: Name: NameFull: Butler, Christopher R. – PersonEntity: Name: NameFull: Mente, Scot – PersonEntity: Name: NameFull: O'Neil, Steven V. – PersonEntity: Name: NameFull: Fonseca, Kari R. – PersonEntity: Name: NameFull: Piro, Justin R. – PersonEntity: Name: NameFull: Cianfrogna, Julie A. – PersonEntity: Name: NameFull: Foley, Timothy L. – PersonEntity: Name: NameFull: Gilbert, Adam M. – PersonEntity: Name: NameFull: Harris, Anthony R. – PersonEntity: Name: NameFull: Helal, Christopher J. – PersonEntity: Name: NameFull: Johnson, Douglas S. – PersonEntity: Name: NameFull: Montgomery, Justin I. – PersonEntity: Name: NameFull: Nason, Deane M. – PersonEntity: Name: NameFull: Noell, Stephen – PersonEntity: Name: NameFull: Pandit, Jayvardhan – PersonEntity: Name: NameFull: Rogers, Bruce N. – PersonEntity: Name: NameFull: Samad, Tarek A. – PersonEntity: Name: NameFull: Shaffer, Christopher L. – PersonEntity: Name: NameFull: Silva, Rafael G. da IsPartOfRelationships: – BibEntity: Dates: – D: 12 M: 04 Text: 4/12/2018 Type: published Y: 2018 Identifiers: – Type: issn-print Value: 00222623 Numbering: – Type: volume Value: 61 – Type: issue Value: 7 Titles: – TitleFull: Journal of Medicinal Chemistry Type: main |
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