Mechanism of the Dual Activities of Human CYP17A1 and Binding to Anti-Prostate Cancer Drug Abiraterone Revealed by a Novel V366M Mutation Causing 17,20 Lyase Deficiency.

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Title: Mechanism of the Dual Activities of Human CYP17A1 and Binding to Anti-Prostate Cancer Drug Abiraterone Revealed by a Novel V366M Mutation Causing 17,20 Lyase Deficiency.
Authors: Fernández-Cancio, Mónica1, Audí, Laura1, Camats, Núria1,2,3, Flück, Christa E.2,3, Zalewski, Adam2,3, Pandey, Amit V.2,3, Dick, Bernhard4, Frey, Brigitte M.4, Monné, Raquel5, Torán, Núria6
Source: Pharmaceuticals (14248247). Jun2018, Vol. 11 Issue 2, p37. 1p.
Database: Academic Search Ultimate
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ISSN:14248247
DOI:10.3390/ph11020037