Development of Kinase Inhibitors via Metal-Catalyzed C-H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies.

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Title: Development of Kinase Inhibitors via Metal-Catalyzed C-H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies.
Authors: Couly, Florence1 florence.couly@insa-rouen.fr, Harari, Marine1 marine.harari@etu.univ-rouen.fr, Dubouilh-Benard, Carole1 carole.dubouilh@univ-rouen.fr, Bailly, Laetitia1 laetitia.bailly@insa-rouen.fr, Petit, Emilie1 emilie.petit@insa-rouen.fr, Diharce, Julien2 julien.diharce@univ-orleans.fr, Bonnet, Pascal2 pascal.bonnet@univ-orleans.fr, Meijer, Laurent3 meijer@manros-therapeutics.com, Fruit, Corinne1 corinne.fruit@univ-rouen.fr, Besson, Thierry1 thierry.besson@univ-rouen.fr
Source: Molecules. Sep2018, Vol. 23 Issue 9, p2181. 16p. 13 Diagrams, 4 Charts.
Database: Academic Search Ultimate
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ISSN:14203049
DOI:10.3390/molecules23092181