Structure-based design and in vivo anti-arthritic activity evaluation of a potent dipeptidyl cyclopropyl nitrile inhibitor of cathepsin C.
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| Title: | Structure-based design and in vivo anti-arthritic activity evaluation of a potent dipeptidyl cyclopropyl nitrile inhibitor of cathepsin C. |
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| Authors: | Korkmaz, Brice1 (AUTHOR) brice.korkmaz@inserm.fr, Lesner, Adam1 (AUTHOR), Wysocka, Magdalena1 (AUTHOR), Gieldon, Artur1 (AUTHOR), Håkansson, Maria1 (AUTHOR), Gauthier, Francis1 (AUTHOR), Logan, Derek T.1 (AUTHOR), Jenne, Dieter E.1 (AUTHOR), Lauritzen, Conni1 (AUTHOR), Pedersen, John1 (AUTHOR) jp@neuprozyme.com |
| Source: | Biochemical Pharmacology. Jun2019, Vol. 164, p349-367. 19p. |
| Database: | Academic Search Ultimate |
| ISSN: | 00062952 |
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| DOI: | 10.1016/j.bcp.2019.04.006 |