Structure-based design and in vivo anti-arthritic activity evaluation of a potent dipeptidyl cyclopropyl nitrile inhibitor of cathepsin C.
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| Title: | Structure-based design and in vivo anti-arthritic activity evaluation of a potent dipeptidyl cyclopropyl nitrile inhibitor of cathepsin C. |
|---|---|
| Authors: | Korkmaz, Brice1 (AUTHOR) brice.korkmaz@inserm.fr, Lesner, Adam1 (AUTHOR), Wysocka, Magdalena1 (AUTHOR), Gieldon, Artur1 (AUTHOR), Håkansson, Maria1 (AUTHOR), Gauthier, Francis1 (AUTHOR), Logan, Derek T.1 (AUTHOR), Jenne, Dieter E.1 (AUTHOR), Lauritzen, Conni1 (AUTHOR), Pedersen, John1 (AUTHOR) jp@neuprozyme.com |
| Source: | Biochemical Pharmacology. Jun2019, Vol. 164, p349-367. 19p. |
| Database: | Academic Search Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: asn DbLabel: Academic Search Ultimate An: 136418205 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=asn&AN=136418205 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bcp.2019.04.006 Languages: – Code: eng Text: English PhysicalDescription: Pagination: PageCount: 19 StartPage: 349 Titles: – TitleFull: Structure-based design and in vivo anti-arthritic activity evaluation of a potent dipeptidyl cyclopropyl nitrile inhibitor of cathepsin C. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Korkmaz, Brice – PersonEntity: Name: NameFull: Lesner, Adam – PersonEntity: Name: NameFull: Wysocka, Magdalena – PersonEntity: Name: NameFull: Gieldon, Artur – PersonEntity: Name: NameFull: Håkansson, Maria – PersonEntity: Name: NameFull: Gauthier, Francis – PersonEntity: Name: NameFull: Logan, Derek T. – PersonEntity: Name: NameFull: Jenne, Dieter E. – PersonEntity: Name: NameFull: Lauritzen, Conni – PersonEntity: Name: NameFull: Pedersen, John IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 06 Text: Jun2019 Type: published Y: 2019 Identifiers: – Type: issn-print Value: 00062952 Numbering: – Type: volume Value: 164 Titles: – TitleFull: Biochemical Pharmacology Type: main |
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